SCHEMBL24716111

SCHEMBL24716111

COc1cccc2c(C3CCNCC3)ccnc12

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.56
HTR1A P08908 10/20 0.54
SLC6A2 P23975 8/20 0.54
SLC6A4 P31645 8/20 0.54
SLC6A3 Q01959 5/20 0.54
JUND P17535 1/20 0.51
FOSB P53539 1/20 0.51
ADRA1D P25100 2/20 0.48
ADRA1A P35348 2/20 0.48
ADRA1B P35368 2/20 0.48
CCNT1 O60563 4/20 0.47
CDK9 P50750 4/20 0.47
HTR6 P50406 1/20 0.43
CDK1 P06493 1/20 0.42
CDK2 P24941 1/20 0.42
CASP3 P42574 1/20 0.42
GSK3B P49841 1/20 0.42
CDK7 P50613 1/20 0.42
CASP7 P55210 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30626631 1.00 HTR2C (0.56) HTR2CHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL25256999 0.87 HTR1A (0.51) HTR2CHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL7967657 0.87 SLC6A2 (0.44) HTR2CHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL24715878 0.86 HTR1A (0.50) HTR2CHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL27196389 0.81 HTR1A (0.47) HTR1ASLC6A2SLC6A4SLC6A3ADRA1D
Hydrochloric Acid SCHEMBL23360080 0.79 HTR1A (0.46) HTR2CHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL30122619 0.78 KMT2A (0.49) HTR1AADRA1DADRA1AADRA1B
SCHEMBL19284730 0.77 HTR2C (0.66) HTR2CHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL30735498 0.77 HTR2C (0.66) HTR2CHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL3693025 0.76 HTR1A (0.51) HTR1AADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4623914-A1 USE OF 8-HYDROXYQUINOLINE DERIVATIVE Jiangsu Yahong Meditech Co., Ltd. (CN) 2025-10-01 EP disclosed
US-20240246916-A1 7-NITRO-8-HYDROXYQUINOLINE DERIVATIVES, PREPARATION METHOD THEREFORE AND MEDICAL USE THEREOF JIANGSU YAHONG MEDITECH CO., LTD. (CN) 2024-07-25 US disclosed
WO-2024109684-A1 USE OF 8-HYDROXYQUINOLINE DERIVATIVE 江苏亚虹医药科技股份有限公司 2024-05-30 WO disclosed
CN-118059101-A Use of 8-hydroxyquinoline derivatives 江苏亚虹医药科技股份有限公司 2024-05-24 CN disclosed
EP-4349815-A1 7-NITRO-8-HYDROXYQUINOLINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF Jiangsu Yahong Meditech Co., Ltd. (CN) 2024-04-10 EP disclosed
CN-117043141-A 7-nitro-8-hydroxyquinoline derivative, preparation method and medical application thereof 江苏亚虹医药科技股份有限公司 2023-11-10 CN disclosed
WO-2022253152-A1 7-NITRO-8-HYDROXYQUINOLINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 江苏亚虹医药科技股份有限公司 2022-12-08 WO disclosed
WO-2022253152-A1 7-NITRO-8-HYDROXYQUINOLINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 江苏亚虹医药科技股份有限公司 2022-12-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240246916-A1 7-NITRO-8-HYDROXYQUINOLINE DERIVATIVES, PREPARATION METHOD THEREFORE AND MEDICAL USE THEREOF CYP3A7, UGT1A7, UGT2B7 HTR2C 1245/4885HTR1A 1797/4885SLC6A2 1212/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.