SCHEMBL2474950

SCHEMBL2474950

C=CCC(N)c1ccccc1-c1nccs1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
PDCD1LG2 Q9BQ51 2/20 0.37
CD274 Q9NZQ7 2/20 0.37
ADRA1A P35348 2/20 0.36
ADRA1D P25100 1/20 0.36
ADRA1B P35368 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.36
FFAR2 O15552 1/20 0.34
RAB9A P51151 2/20 0.33
ADRA2A P08913 1/20 0.33
CYP2A6 P11509 1/20 0.33
HSP90AA1 P07900 1/20 0.32
CASP6 P55212 1/20 0.32
TGFBR1 P36897 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
NPC1 O15118 1/20 0.31
ADRB2 P07550 1/20 0.31
F2RL1 P55085 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8145857 0.76 PDPK1 (0.46) PDPK1ADORA2AADORA1ADRA1AADRA1D
SCHEMBL2480653 0.75 LTA4H (0.39) ADORA2AADORA1PDCD1LG2CD274RAB9A
SCHEMBL27763732 0.72 PDPK1 (0.42) PDPK1ADORA2AADORA1ADRA1AADRA1D
SCHEMBL10044886 0.72 PDPK1 (0.48) PDPK1ADORA2AADORA1ADRA1AADRA1D
Hydrochloric Acid SCHEMBL2474756 0.72 KDM4E (0.50) PDCD1LG2CD274RAB9ANPC1
SCHEMBL3105786 0.71 PTPRC (0.37) PDCD1LG2CD274ADRA1AADRA1DADRA1B
Hydrochloric Acid SCHEMBL2480213 0.71 PDCD1LG2 (0.39) PDCD1LG2CD274RAB9ACYP2A6ADRB2
SCHEMBL5692672 0.71 PDPK1 (0.64) PDPK1ADORA2AADORA1ADRA1AADRA1D
SCHEMBL2477497 0.70 PDCD1LG2 (0.39) PDCD1LG2CD274
SCHEMBL2473298 0.70 PDCD1LG2 (0.44) PDCD1LG2CD274RAB9ACYP2A6NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2159216-B1 3-BUTENYL-1-AMINE DERIVATIVES AND THEIR USE AS Ih MODULORS FOR THE TREATMENT OF PSYCHIATIRC DISORDERS ORGANON NV (NL) 2011-10-12 EP disclosed
EP-2159216-A1 Ih - Modulators N.V. Organon (NL) 2010-03-03 EP disclosed
US-20020037885-A1 Therapeutic compounds DIJCKS FREDERICUS ANTONIUS (NL) 2002-03-28 US disclosed
US-6313139-B1 ADMINISTERING BENZYLAMINE DERIVATIVE FOR THERAPY OF PSYCHIATRIC DISORDER IN MAMMALS AKZO NOBEL N. V. (NL) 2001-11-06 US disclosed
EP-1035843-A2 I h?-MODULATORS Akzo Nobel N.V. (NL) 2000-09-20 EP disclosed
US-6080773-A USEFUL FOR TREATMENT OF DEPRESSION, ANXIETY OR PSYCHOSIS AKZO NOBEL, N.V. (NL) 2000-06-27 US disclosed
WO-1999018941-A2 Ih-MODULATORS AKZO NOBEL N.V. (NL) 1999-04-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020037885-A1 Therapeutic compounds BDNF, PNMT, SLC18A2 PDPK1 1216/4885ADORA2A 71/4885ADORA1 229/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.