SCHEMBL24767003

SCHEMBL24767003

COc1cc(Br)ccc1OCC1CO1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
GLA P06280 1/20 0.49
DRD4 P21917 5/20 0.48
TP53 P04637 1/20 0.44
CYP3A4 P08684 1/20 0.44
TSHR P16473 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HIF1A Q16665 1/20 0.44
ADRA2C P18825 1/20 0.43
TDP1 Q9NUW8 2/20 0.42
KDM4E B2RXH2 1/20 0.42
PKM P14618 1/20 0.41
PTPN1 P18031 1/20 0.41
SLC6A4 P31645 1/20 0.41
PYGL P06737 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28343422 0.89 DRD4 (0.48) ALDH1A1DRD4ADRA2CKDM4E
SCHEMBL20203110 0.89 DRD4 (0.48) ALDH1A1DRD4ADRA2CKDM4E
SCHEMBL29847833 0.84 ALDH1A1 (0.60) ALDH1A1GLADRD4TP53CYP3A4
SCHEMBL25812948 0.83 CA12 (0.53) ALDH1A1GLADRD4TP53CYP3A4
SCHEMBL7966936 0.83 ALDH1A1 (0.54) ALDH1A1GLATP53CYP3A4TSHR
SCHEMBL16923006 0.83 ALDH1A1 (0.57) ALDH1A1GLADRD4TP53CYP3A4
SCHEMBL7966930 0.83 ALDH1A1 (0.54) ALDH1A1GLATP53CYP3A4TSHR
SCHEMBL7966929 0.83 ALDH1A1 (0.54) ALDH1A1GLATP53CYP3A4TSHR
SCHEMBL28343556 0.82 DRD4 (0.41) ALDH1A1DRD4TDP1KDM4ESLC6A4
SCHEMBL4892470 0.82 ALDH1A1 (0.49) ALDH1A1GLATP53CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115385847-B Polysubstituted diaryl compound, preparation method and application thereof 山东第一医科大学(山东省医学科学院) 2023-09-29 CN disclosed
WO-2022262350-A1 SUBSTITUTED DIARYL COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 山东第一医科大学(山东省医学科学院) 2022-12-22 WO disclosed
CN-115385847-A Polysubstituted diaryl compound and preparation method and application thereof 山东第一医科大学(山东省医学科学院) 2022-11-25 CN disclosed
CN-113387873-B Substituted diaryl compound, preparation method and application thereof 山东第一医科大学(山东省医学科学院) 2022-09-20 CN disclosed