SCHEMBL24767809

SCHEMBL24767809

COC(=O)c1ccc(-n2cccc2)c(N)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.61
NPC1 O15118 3/20 0.61
RAB9A P51151 2/20 0.61
NPSR1 Q6W5P4 2/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
ALDH1A1 P00352 8/20 0.57
HPGD P15428 6/20 0.57
MAPT P10636 6/20 0.57
GAA P10253 4/20 0.57
HSD17B10 Q99714 3/20 0.57
GLA P06280 1/20 0.57
CASP1 P29466 1/20 0.57
CASP7 P55210 1/20 0.57
ATM Q13315 1/20 0.57
PKM P14618 2/20 0.49
USP2 O75604 1/20 0.49
LMNA P02545 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
ALOX15 P16050 1/20 0.46
MAPK1 P28482 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3793807 0.84 PRMT1 (0.57) KDM4ENPC1RAB9ANPSR1SMN1; SMN2
SCHEMBL31213036 0.83 CA12 (0.59) KDM4ENPC1RAB9ANPSR1SMN1; SMN2
SCHEMBL2592774 0.83 CA12 (0.59) KDM4ENPC1RAB9ANPSR1SMN1; SMN2
SCHEMBL9692785 0.81 HTT (0.62) KDM4ENPC1RAB9ANPSR1SMN1; SMN2
SCHEMBL29171465 0.80 KDM4E (0.57) KDM4ENPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL11355898 0.80 KDM4E (0.44) KDM4ENPC1RAB9ANPSR1SMN1; SMN2
SCHEMBL7827414 0.79 ALDH1A1 (0.53) KDM4ENPC1RAB9ANPSR1SMN1; SMN2
SCHEMBL27469088 0.79 ALDH1A1 (0.59) KDM4ENPC1RAB9ANPSR1SMN1; SMN2
SCHEMBL7823115 0.79 CA12 (0.59) KDM4ESMN1; SMN2ALDH1A1HPGDMAPT
SCHEMBL16869458 0.79 KDM4E (0.54) KDM4ENPC1RAB9ANPSR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118184632-A Pyrrolo [1,2-a ] quinoxaline compound synthesized from aminopyrrole arene and carbon dioxide and synthesis method thereof 陕西科技大学 2024-06-14 CN claimed
US-20240262812-A1 N-SUBSTITUTED PHENYLSULFONAMIDE COMPOUND AND USE THEREOF SHANGHAI LEADO PHARMATECH CO. LTD. (CN) 2024-08-08 US disclosed
CN-115477626-B N-substituted phenyl sulfonamide compound and application thereof 上海璃道医药科技有限公司 2024-08-02 CN disclosed
CN-118184632-A Pyrrolo [1,2-a ] quinoxaline compound synthesized from aminopyrrole arene and carbon dioxide and synthesis method thereof 陕西科技大学 2024-06-14 CN disclosed
EP-4357338-A1 N-SUBSTITUTED PHENYLSULFONAMIDE COMPOUND AND USE THEREOF Shanghai Leado Pharmatech Co. Ltd. (CN) 2024-04-24 EP disclosed
CN-117529474-A N-substituted phenyl sulfonamide compound and application thereof 上海璃道医药科技有限公司 2024-02-06 CN disclosed
WO-2022262657-A1 N-SUBSTITUTED PHENYLSULFONAMIDE COMPOUND AND USE THEREOF 上海璃道医药科技有限公司 2022-12-22 WO disclosed
WO-2022262657-A1 N-SUBSTITUTED PHENYLSULFONAMIDE COMPOUND AND USE THEREOF 上海璃道医药科技有限公司 2022-12-22 WO disclosed
CN-115477626-A N-substituted phenylsulfonamide compound and application thereof 上海璃道医药科技有限公司 2022-12-16 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240262812-A1 N-SUBSTITUTED PHENYLSULFONAMIDE COMPOUND AND USE THEREOF TRPV1, TRPA1, TRPV5 KDM4E 2673/4885NPC1 1827/4885RAB9A 1135/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.