SCHEMBL2477934

SCHEMBL2477934

O=C1CC(F)(c2ccccc2)Oc2ccccc21

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.45
ATM Q13315 1/20 0.43
CFTR P13569 1/20 0.42
GOPC Q9HD26 1/20 0.42
MAOB P27338 3/20 0.39
KDM4E B2RXH2 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
AR P10275 1/20 0.39
CYP19A1 P11511 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HSD11B1 P28845 1/20 0.38
EPHX2 P34913 2/20 0.37
CYP2C9 P11712 1/20 0.37
ADRA1D P25100 2/20 0.36
ADRA1A P35348 2/20 0.36
ADRA1B P35368 2/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11256545 0.79 SIGMAR1 (0.47) SIGMAR1ATMCFTRGOPCMAOB
SCHEMBL6704259 0.79 SIGMAR1 (0.47) SIGMAR1ATMCFTRGOPCMAOB
SCHEMBL29818629 0.79 SIGMAR1 (0.47) SIGMAR1ATMCFTRGOPCMAOB
SCHEMBL30499348 0.79 KDM4E (0.57) MAOBKDM4EARCYP19A1HSD17B10
SCHEMBL31190168 0.77 SIGMAR1 (0.45) SIGMAR1ATMCFTRGOPCMAOB
SCHEMBL1534682 0.77 SIGMAR1 (0.45) SIGMAR1ATMCFTRGOPCMAOB
SCHEMBL2022537 0.77 SIGMAR1 (0.45) SIGMAR1ATMCFTRGOPCMAOB
SCHEMBL927371 0.77 SIGMAR1 (0.45) SIGMAR1ATMCFTRGOPCMAOB
SCHEMBL9278695 0.77 ATM (0.47) SIGMAR1ATMCFTRGOPCMAOB
SCHEMBL753626 0.77 SIGMAR1 (0.45) SIGMAR1ATMCFTRGOPCMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376408-A2 FLUORINATION OF ORGANIC COMPOUNDS President and Fellows of Harvard College (US) 2011-10-19 EP claimed
WO-2010059943-A2 FLUORINATION OF ORGANIC COMPOUNDS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-05-27 WO claimed
US-5399584-A Preventing gastrointestinal damage caused by nonsteroidal antiinflammatory drugs THE PROCTER & GAMBLE COMPANY (US) 1995-03-21 US claimed
US-5399584-A Preventing gastrointestinal damage caused by nonsteroidal antiinflammatory drugs THE PROCTER & GAMBLE COMPANY (US) 1995-03-21 US disclosed