SCHEMBL24802438

SCHEMBL24802438

Cc1cnc(O)c(N2CCN(C)C2=O)c1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.36
SCN10A Q9Y5Y9 1/20 0.36
CYP11B2 P19099 1/20 0.34
PIM1 P11309 1/20 0.33
PDE10A Q9Y233 1/20 0.32
PARP1 P09874 1/20 0.32
CYP17A1 P05093 1/20 0.30
NTRK1 P04629 1/20 0.30
LCK P06239 1/20 0.30
KDR P35968 1/20 0.30
JAK3 P52333 1/20 0.30
MAPK14 Q16539 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30
NOS2 P35228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24802440 0.79 CYP17A1 (0.37) SCN9ASCN10ACYP11B2PIM1PDE10A
SCHEMBL26449823 0.70 GRM5 (0.42) PDE10ANOS3NOS2
SCHEMBL23416642 0.66 GAA (0.35) NOS3NOS1NOS2
SCHEMBL22542026 0.66 SCN9A (0.43) SCN9ASCN10APARP1NTRK1
SCHEMBL24804886 0.65 SCN9A (0.35) SCN9ASCN10ACYP11B2PIM1PARP1
SCHEMBL30772165 0.65 SCN9A (0.35) SCN9ASCN10ACYP11B2PIM1PARP1
SCHEMBL11493940 0.65 HSD17B10 (0.41) SCN9ASCN10APARP1
SCHEMBL12362742 0.65 CA12 (0.38) SCN9ASCN10APARP1KDR
SCHEMBL30148626 0.65 RAF1 (0.38)
SCHEMBL27774656 0.64 PIM1 (0.39) SCN9ASCN10APIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022268209-A1 DERIVATIVE HAVING PYRIMIDINE-FUSED CYCLIC STRUCTURE, AND USE THEREOF 四川汇宇制药股份有限公司 2022-12-29 WO disclosed