SCHEMBL30148626

SCHEMBL30148626

COc1ncc(NC(=O)O)cc1N1CCN(C)C1=O

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 10/20 0.38
BRAF P15056 10/20 0.38
MALT1 Q9UDY8 3/20 0.37
HTR2A P28223 3/20 0.36
HTR2C P28335 3/20 0.36
HTR2B P41595 3/20 0.36
BACE1 P56817 1/20 0.35
PRMT5 O14744 1/20 0.32
WDR77 Q9BQA1 1/20 0.32
SLC13A5 Q86YT5 2/20 0.32
SLC13A2 Q13183 1/20 0.32
SLC13A3 Q8WWT9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29180862 0.85 RORC (0.42) RAF1BRAFMALT1BACE1
SCHEMBL30772208 0.85 RORC (0.42) RAF1BRAFMALT1BACE1
Hydrochloric Acid SCHEMBL29180786 0.84 CYP17A1 (0.33) RAF1BRAFMALT1
SCHEMBL24802440 0.81 CYP17A1 (0.37) SLC13A5SLC13A2SLC13A3
SCHEMBL30772165 0.78 SCN9A (0.35) RAF1
SCHEMBL24804886 0.78 SCN9A (0.35) RAF1
SCHEMBL30148717 0.77 ALDH1A1 (0.34)
SCHEMBL29180832 0.76 CYP11B2 (0.35)
SCHEMBL22574269 0.74 CYP11B2 (0.45) PRMT5WDR77
SCHEMBL30772189 0.73 KAT2B (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022268209-A1 DERIVATIVE HAVING PYRIMIDINE-FUSED CYCLIC STRUCTURE, AND USE THEREOF 四川汇宇制药股份有限公司 2022-12-29 WO disclosed