SCHEMBL24802440

SCHEMBL24802440

COc1ncc(C)cc1N1CCN(C)C1=O

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 4/20 0.37
SCN9A Q15858 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.35
PIM1 P11309 1/20 0.34
SLC13A5 Q86YT5 2/20 0.34
SLC13A2 Q13183 1/20 0.34
SLC13A3 Q8WWT9 1/20 0.34
CRHR1 P34998 1/20 0.34
CCR9 P51686 1/20 0.33
KAT2B Q92831 1/20 0.32
PIK3CD O00329 3/20 0.31
PIK3CA P42336 1/20 0.31
MTOR P42345 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
PDE10A Q9Y233 1/20 0.31
PARP1 P09874 1/20 0.31
CYP11B2 P19099 1/20 0.31
SSTR4 P31391 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30772165 0.86 SCN9A (0.35) CYP17A1SCN9ASCN10APIM1CRHR1
SCHEMBL24804886 0.86 SCN9A (0.35) CYP17A1SCN9ASCN10APIM1CRHR1
Hydrochloric Acid SCHEMBL29180786 0.81 CYP17A1 (0.33) CYP17A1SCN9ASCN10APIM1CRHR1
SCHEMBL30148626 0.81 RAF1 (0.38) SLC13A5SLC13A2SLC13A3
SCHEMBL30772189 0.80 KAT2B (0.37) CYP17A1SCN9ASCN10AKAT2B
SCHEMBL24802438 0.79 SCN9A (0.36) CYP17A1SCN9ASCN10APIM1HRH3
SCHEMBL29180832 0.78 CYP11B2 (0.35) CYP17A1SCN9ASCN10APIM1CRHR1
SCHEMBL46303 0.77 HSD17B10 (0.46) CYP11B2
SCHEMBL30148717 0.76 ALDH1A1 (0.34) PIK3CDHRH3
SCHEMBL29180830 0.74 SCN9A (0.33) SCN9ASCN10ACRHR1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022268209-A1 DERIVATIVE HAVING PYRIMIDINE-FUSED CYCLIC STRUCTURE, AND USE THEREOF 四川汇宇制药股份有限公司 2022-12-29 WO disclosed