SCHEMBL2480466

SCHEMBL2480466

CC(C#N)(C(=O)O)C1(C[N+](=O)[O-])C(=O)Nc2ccc(Cl)cc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.42
CBX7 O95931 2/20 0.37
CDYL Q9Y232 2/20 0.37
CDYL2 Q8N8U2 1/20 0.37
CDY1; CDY1B Q9Y6F8 1/20 0.37
MGAM O43451 1/20 0.35
HTR1A P08908 1/20 0.35
GAA P10253 1/20 0.35
SI P14410 1/20 0.35
HTR2A P28223 1/20 0.35
HTR7 P34969 1/20 0.35
HTR6 P50406 1/20 0.35
MGAM2 Q2M2H8 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
BCHE P06276 1/20 0.34
MDM2 Q00987 4/20 0.33
IP6K1 Q92551 2/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16377143 0.73 IDO1 (0.62) IDO1CBX7CDYLCDYL2CDY1; CDY1B
SCHEMBL2485622 0.72 IDO1 (0.41) IDO1CBX7CDYLCDYL2CDY1; CDY1B
SCHEMBL2482415 0.72 PGR (0.41) IDO1CBX7CDYLCDYL2CDY1; CDY1B
SCHEMBL2485480 0.70 MDM2 (0.38) IDO1MDM2TP53AKR1B1
SCHEMBL11959125 0.69 IDO1 (0.41) IDO1CBX7CDYLCDYL2CDY1; CDY1B
SCHEMBL2485481 0.68 IDO1 (0.48) IDO1CBX7CDYLCDYL2CDY1; CDY1B
SCHEMBL12205319 0.66 PGR (0.43) IDO1CBX7CDYLCDYL2CDY1; CDY1B
SCHEMBL12205346 0.65 IDO1 (0.43) IDO1CBX7CDYLCDYL2CDY1; CDY1B
SCHEMBL9542686 0.61 ADAM17 (0.48) BCHEAKR1B1
SCHEMBL1722012 0.59 PGR (0.69) IDO1MEN1KMT2AAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891075-B1 TRICYCLIC SPIRO DERIVATIVES AS CRTH2 MODULATORS MERCK SERONO SA (CH) 2011-10-19 EP disclosed