SCHEMBL24808653

SCHEMBL24808653

Cc1cc(F)cc(N(CC(F)(F)F)c2nc(=O)[nH]c3cc(Cl)ccc23)c1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAT2A P31153 7/20 0.52
TP53 P04637 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
LMNA P02545 1/20 0.35
HAVCR2 Q8TDQ0 1/20 0.34
AR P10275 4/20 0.33
NOS2 P35228 1/20 0.33
CHEK1 O14757 1/20 0.33
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24808651 0.88 MAT2A (0.49) MAT2ATP53SMN1; SMN2LMNAHAVCR2
SCHEMBL24807300 0.85 AR (0.40) SMN1; SMN2LMNAAR
SCHEMBL24807294 0.80 MAT2A (0.41) MAT2A
SCHEMBL24807286 0.79 MAT2A (0.50) MAT2AARNOS2
SCHEMBL24807057 0.76 MAT2A (0.51) MAT2ATP53SMN1; SMN2LMNAHAVCR2
SCHEMBL23601671 0.74 MAT2A (0.30) MAT2A
SCHEMBL24807047 0.72 MAT2A (0.62) MAT2ATP53SMN1; SMN2LMNAHAVCR2
SCHEMBL24807299 0.72 AR (0.35) AR
SCHEMBL30095575 0.72 AR (0.35) AR
SCHEMBL24807042 0.71 MAT2A (0.41) MAT2ANOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230060004-A1 DIACYLGLYERCOL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2023-02-23 US disclosed
WO-2022271677-A1 DIACYLGLYERCOL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2022-12-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230060004-A1 DIACYLGLYERCOL KINASE MODULATING COMPOUNDS DGKG, DGKB, DGKK MAT2A 1466/4885TP53 817/4885SMN1; SMN2 4820/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.