SCHEMBL24809118

SCHEMBL24809118

C[Si](C)(C)CCOCn1nc(-c2ccncc2)c2cc(Br)ccc21

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.40
MAPK14 Q16539 1/20 0.34
KMT2A Q03164 1/20 0.33
NAMPT P43490 4/20 0.33
NPC1 O15118 1/20 0.32
MAPT P10636 2/20 0.32
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
DYRK1A Q13627 1/20 0.30
SLC6A2 P23975 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16014263 0.87 DGAT1 (0.43) DGAT1NPC1DYRK1A
SCHEMBL30084147 0.86 NPC1 (0.34) DGAT1MAPK14NAMPTNPC1MAPT
SCHEMBL3515565 0.86 NPC1 (0.34) DGAT1MAPK14NAMPTNPC1MAPT
SCHEMBL17432551 0.86 DGAT1 (0.39) DGAT1NPC1MAPTDYRK1A
SCHEMBL14493396 0.85 MKNK1 (0.41) MAPK14KMT2ANPC1MAPTALDH1A1
SCHEMBL3515950 0.82 L3MBTL1 (0.47) NPC1MAPT
SCHEMBL23783005 0.81 DGAT1 (0.40) DGAT1KMT2ANAMPTNPC1CYP3A4
SCHEMBL757561 0.81 DGAT1 (0.38) DGAT1KMT2ANPC1MAPTALDH1A1
SCHEMBL16024590 0.81 DGAT1 (0.38) DGAT1MAPK14
SCHEMBL30084198 0.81 MAPT (0.37) MAPK14KMT2ANAMPTNPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022271840-A1 SELECTIVE INDAZOLE LRRK2 INHIBITORS AND METHODS FOR USE THEREOF THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2022-12-29 WO disclosed
WO-2022271840-A1 SELECTIVE INDAZOLE LRRK2 INHIBITORS AND METHODS FOR USE THEREOF THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2022-12-29 WO disclosed