SCHEMBL2483209

SCHEMBL2483209

COc1ccc(N)cc1N1CCOCC1.COc1ccc([N+](=O)[O-])cc1N1CCOCC1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A5 Q9Y345 3/20 0.55
MAPK1 P28482 2/20 0.52
HTT P42858 2/20 0.52
PAX8 Q06710 1/20 0.52
ALDH1A1 P00352 4/20 0.51
RAB9A P51151 2/20 0.51
MITF O75030 1/20 0.51
LMNA P02545 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
MAPT P10636 1/20 0.50
HSP90AA1 P07900 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
SLC6A9 P48067 2/20 0.48
KMT2A Q03164 3/20 0.48
MEN1 O00255 1/20 0.47
PKM P14618 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29833031 0.93 SLC6A5 (0.61) SLC6A5MAPK1HTTPAX8ALDH1A1
SCHEMBL520263 0.93 SLC6A5 (0.61) SLC6A5MAPK1HTTPAX8ALDH1A1
SCHEMBL29833266 0.86 MAPT (0.57) ALDH1A1RAB9ALMNASMN1; SMN2MAPT
SCHEMBL519902 0.86 MAPT (0.57) ALDH1A1RAB9ALMNASMN1; SMN2MAPT
SCHEMBL29788533 0.82 SLC6A5 (0.64) SLC6A5MAPK1HTTPAX8ALDH1A1
SCHEMBL2062084 0.82 SLC6A5 (0.64) SLC6A5MAPK1HTTPAX8ALDH1A1
SCHEMBL12528187 0.81 SLC6A5 (0.63) SLC6A5MAPK1HTTPAX8ALDH1A1
SCHEMBL10035015 0.80 ALDH1A1 (0.52) SLC6A5MAPK1HTTPAX8ALDH1A1
SCHEMBL3252580 0.79 ALDH1A1 (0.63) MAPK1HTTPAX8ALDH1A1RAB9A
SCHEMBL4865184 0.78 HTR6 (0.62) MAPK1HTTALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376491-A1 PYRROLOTRIAZINES AS ALK AND JAK2 INHIBITORS Cephalon, Inc. (US) 2011-10-19 EP disclosed
WO-2010071885-A1 PYRROLOTRIAZINES AS ALK AND JAK2 INHIBITORS CEPHALON, INC. (US) 2010-06-24 WO disclosed