SCHEMBL2483754

SCHEMBL2483754

O=[C]c1ccc([N+](=O)[O-])c([N+](=O)[O-])c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.52
CYP3A4 P08684 4/20 0.52
VCAM1 P19320 2/20 0.47
CASP6 P55212 1/20 0.47
TDP1 Q9NUW8 6/20 0.41
MAPK1 P28482 2/20 0.41
ATM Q13315 1/20 0.41
GPR35 Q9HC97 1/20 0.39
ALDH1A1 P00352 3/20 0.38
MAPT P10636 3/20 0.38
CYP1A2 P05177 2/20 0.38
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
GRIK1 P39086 1/20 0.38
GRIA1 P42261 1/20 0.38
GRIA2 P42262 1/20 0.38
GRIA3 P42263 1/20 0.38
GRIA4 P48058 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11673788 0.83 TSHR (0.44) TSHRCYP3A4VCAM1CASP6TDP1
SCHEMBL7734099 0.83 VCAM1 (0.44) TSHRCYP3A4VCAM1TDP1MAPK1
SCHEMBL7153973 0.82 GPR35 (0.58) TSHRCYP3A4VCAM1TDP1MAPK1
SCHEMBL697848 0.82 ALDH1A1 (0.58) VCAM1CASP6TDP1ATMALDH1A1
SCHEMBL5163347 0.82 TSHR (0.56) TSHRCYP3A4VCAM1TDP1MAPK1
SCHEMBL7151564 0.82 MAPK1 (0.58) TSHRCYP3A4VCAM1MAPK1GPR35
SCHEMBL10348032 0.82 TSHR (0.60) TSHRCYP3A4VCAM1TDP1MAPK1
SCHEMBL698857 0.82 VCAM1 (0.71) TSHRVCAM1TDP1MAPK1MAPT
SCHEMBL29217568 0.82 TDP1 (0.60) TSHRCYP3A4VCAM1TDP1MAPK1
SCHEMBL27799226 0.82 MAPT (0.60) TSHRCYP3A4VCAM1TDP1GPR35

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1035614-C Benzylidene derivatives SHIONOGI & CO (JP) 1997-08-13 CN claimed
EP-0595546-B1 Benzylidene derivatives SHIONOGI & CO (JP) 1996-03-20 EP claimed
US-5418230-A Antiinflammatory SHIONOGI & CO., LTD. (JP) 1995-05-23 US claimed
US-4472386-A 5-Fluoro-(β-uridine or 2'-deoxy-β-uridine) derivatives, a process for producing the same and a carcinostatic agent containing the same TOYAMA CHEMICAL CO., LTD. (JP) 1984-09-18 US claimed
CN-110577489-B Synthetic method of narcotic analgesic 宜昌人福药业有限责任公司 2023-02-21 CN disclosed
CN-112079823-B Near-infrared frequency up-conversion fluorescence molecular probe, preparation method and application 中国药科大学 2022-03-29 CN disclosed
CN-112079823-A Near-infrared frequency up-conversion fluorescence molecular probe, preparation method and application 中国药科大学 2020-12-15 CN disclosed
CN-110577489-A Synthetic method of narcotic analgesic 宜昌人福药业有限责任公司 2019-12-17 CN disclosed
US-9045520-B2 Synthesis of purine nucleosides GILEAD PHARMASSET LLC (US) 2015-06-02 US disclosed
CN-104557472-A Adamantane derivative, preparation method and application in epoxy resin UNIV BEIJING CHEMICAL 2015-04-29 CN disclosed
US-8716263-B2 Synthesis of purine nucleosides GILEAD PHARMASSET LLC (US) 2014-05-06 US disclosed
EP-2671888-A1 3',5'-cyclic nucleoside phosphate analogues Gilead Pharmasset LLC (US) 2013-12-11 EP disclosed
US-6114566-A 4-cyano-3-hydroxybutanoyl hydrazines, derivatives and process for the preparation thereof BOARD OF TRUSTEES OPERATING MICHIGAN STATE UNIVERSITY (US) 2000-09-05 US disclosed
EP-1026162-A1 ANTIRHEUMATIC SHIONOGI & CO., LTD. (JP) 2000-08-09 EP disclosed
CN-1035614-C Benzylidene derivatives SHIONOGI & CO (JP) 1997-08-13 CN disclosed
EP-0595546-B1 Benzylidene derivatives SHIONOGI & CO (JP) 1996-03-20 EP disclosed
CN-1092414-A Benzylidene derivatives SHIONOGI & CO (JP) 1994-09-21 CN disclosed
EP-0595546-A1 Benzylidene derivatives SHIONOGI & CO., LTD. (JP) 1994-05-04 EP disclosed
US-4472386-A 5-Fluoro-(β-uridine or 2'-deoxy-β-uridine) derivatives, a process for producing the same and a carcinostatic agent containing the same TOYAMA CHEMICAL CO., LTD. (JP) 1984-09-18 US disclosed
EP-0092830-A2 Cephalosporin derivatives, process for their preparation, pharmaceutical compositions containing them and their application CIBA-GEIGY AG (CH) 1983-11-02 EP disclosed