SCHEMBL2484185

SCHEMBL2484185

CCCCOc1cccc2cccnc12

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.68
KDM4E B2RXH2 5/20 0.68
LMNA P02545 5/20 0.68
RAB9A P51151 4/20 0.68
NPC1 O15118 3/20 0.68
SMN1; SMN2 Q16637 3/20 0.68
MEN1 O00255 2/20 0.68
KMT2A Q03164 2/20 0.68
GAA P10253 1/20 0.68
CYP1A2 P05177 1/20 0.65
CYP3A4 P08684 1/20 0.65
CYP2D6 P10635 1/20 0.65
CYP2C19 P33261 1/20 0.65
MCHR1 Q99705 2/20 0.65
POLB P06746 1/20 0.64
ALDH1A1 P00352 1/20 0.61
HPGD P15428 1/20 0.61
MAPK1 P28482 1/20 0.61
HTT P42858 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9568616 0.95 MAPT (0.66) MAPTKDM4ELMNARAB9ANPC1
SCHEMBL9632939 0.93 MCHR1 (0.67) MAPTKDM4ELMNARAB9ANPC1
SCHEMBL16114005 0.93 MCHR1 (0.67) MAPTKDM4ELMNARAB9ANPC1
SCHEMBL18691791 0.93 MCHR1 (0.67) MAPTKDM4ELMNARAB9ANPC1
SCHEMBL10647335 0.93 MCHR1 (0.67) MAPTKDM4ELMNARAB9ANPC1
SCHEMBL2484526 0.91 MAPT (0.66) MAPTKDM4ELMNARAB9ANPC1
SCHEMBL19733316 0.87 MCHR1 (0.58) MAPTKDM4ELMNARAB9ANPC1
SCHEMBL2485359 0.85 RAB9A (0.75) MAPTKDM4ELMNARAB9ANPC1
SCHEMBL30982342 0.84 RAB9A (0.71) MAPTKDM4ELMNARAB9ANPC1
SCHEMBL10460812 0.84 RAB9A (0.71) MAPTKDM4ELMNARAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100376604-C Olefin polymerization catalyst and its uses CHINA PETROLEUM & CHEMICAL (CN) 2008-03-26 CN claimed
CN-1769307-A Olefin polymerization catalyst and its uses CHINA PETROLEUM & CHEMICAL (CN) 2006-05-10 CN claimed
WO-2017094872-A1 ULTRAVIOLET ABSORBER 国立大学法人大阪大学 2017-06-08 WO disclosed
US-8013153-B2 Substituted pyrimidine kinase inhibitors JANSSEN PHARMACEUTICA, N.V. (BE) 2011-09-06 US disclosed
CN-100376604-C Olefin polymerization catalyst and its uses CHINA PETROLEUM & CHEMICAL (CN) 2008-03-26 CN disclosed
US-20070254896-A1 SUBSTITUTED PYRIMIDINE KINASE INHIBITORS JANSSEN PHARMACEUTICA, N.V. (BE) 2007-11-01 US disclosed
CN-1769307-A Olefin polymerization catalyst and its uses CHINA PETROLEUM & CHEMICAL (CN) 2006-05-10 CN disclosed
US-5405843-A Anticancer drug potentiators MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1995-04-11 US disclosed
EP-0435687-B1 Process for isomerization of oxime ethers SUMITOMO CHEMICAL CO (JP) 1995-03-29 EP disclosed
EP-0363212-B1 Novel heterocyclic compounds and anticancer-drug reinforcing agents containing them as effective components MITSUI TOATSU CHEMICALS (JP) 1995-01-04 EP disclosed
EP-0428351-B1 Synthesis of quinoline and substituted quinoline copolymers EXXON RESEARCH ENGINEERING CO (US) 1994-12-21 EP disclosed
US-5204348-A Quinoline derivatives MITSUI TOATSU CHEMICALS INC. (JP) 1993-04-20 US disclosed
US-5162495-A Contacting tetrahydroquinoline compound with a quinoline compound in presence of metal sulfide catalyst EXXON RESEARCH AND ENGINEERING COMPANY (US) 1992-11-10 US disclosed
US-5130486-A A ketoximine ether isomerized using a Lewis acid metal halide SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1992-07-14 US disclosed
US-5112817-A Anticancer Drug Potentiators MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1992-05-12 US disclosed
EP-0435687-A2 Process for isomerization of oxime ethers SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1991-07-03 EP disclosed
EP-0428351-A2 Synthesis of quinoline and substituted quinoline copolymers EXXON RESEARCH AND ENGINEERING COMPANY (US) 1991-05-22 EP disclosed
EP-0363212-A2 Novel heterocyclic compounds and anticancer-drug reinforcing agents containing them as effective components MITSUI TOATSU CHEMICALS, Inc. (JP) 1990-04-11 EP disclosed
US-4031215-A STREPTOMYCES, ALDOL CONDENSATION KAKEN CHEMICAL CO., LTD. (JA) 1977-06-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070254896-A1 SUBSTITUTED PYRIMIDINE KINASE INHIBITORS DTYMK, TK1, DCK MAPT 2869/4885KDM4E 2150/4885LMNA 3668/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.