SCHEMBL24865172

SCHEMBL24865172

Cc1cc(N2CCC(C(F)(F)F)CC2)ccc1Nc1ccc2oc(=O)[nH]c2c1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 13/20 0.41
JAK3 P52333 13/20 0.41
JAK2 O60674 7/20 0.41
CYP3A4 P08684 5/20 0.41
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
CYP1A2 P05177 1/20 0.36
TYK2 P29597 1/20 0.36
P2RX3 P56373 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31123300 1.00 JAK1 (0.41) JAK1JAK3JAK2CYP3A4NOS3
SCHEMBL24865555 0.93 MEN1 (0.39)
SCHEMBL31123262 0.93 MEN1 (0.39)
SCHEMBL24865673 0.87 JAK1 (0.41) JAK1JAK3JAK2CYP3A4NOS3
SCHEMBL31123276 0.87 JAK1 (0.41) JAK1JAK3JAK2CYP3A4NOS3
SCHEMBL24865446 0.84 BCL6 (0.39) JAK2
SCHEMBL31123302 0.84 BCL6 (0.39) JAK2
SCHEMBL24864899 0.76 ADRB1 (0.33)
SCHEMBL24865460 0.76 TRPV1 (0.59)
SCHEMBL24865324 0.76 TRPV1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117999259-A Iron death modulators, their preparation and use 维泰瑞隆有限公司 2024-05-07 CN disclosed
WO-2023280296-A1 FERROPTOSIS MODULATORS, PREPARATIONS, AND USES THEREOF Sironax Ltd. (KY) 2023-01-12 WO disclosed