SCHEMBL24865446

SCHEMBL24865446

Cc1cc(N2CCC(C(F)(F)F)CC2)ccc1Nc1ccc2[nH]c(=O)[nH]c2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL6 P41182 7/20 0.39
BCOR Q6W2J9 7/20 0.39
KMT2A Q03164 4/20 0.36
MEN1 O00255 3/20 0.36
JAK2 O60674 1/20 0.36
SYK P43405 1/20 0.36
MAPT P10636 4/20 0.36
POLB P06746 2/20 0.36
TSHR P16473 1/20 0.36
CASP1 P29466 1/20 0.36
HBB P68871 1/20 0.36
ALDH1A1 P00352 4/20 0.36
GAA P10253 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PDE3B Q13370 2/20 0.35
PDE3A Q14432 2/20 0.35
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
HTR2A P28223 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31123302 1.00 BCL6 (0.39) BCL6BCORKMT2AMEN1JAK2
SCHEMBL31123262 0.84 MEN1 (0.39) KMT2AMEN1
SCHEMBL31123300 0.84 JAK1 (0.41) JAK2
SCHEMBL24865555 0.84 MEN1 (0.39) KMT2AMEN1
SCHEMBL24865172 0.84 JAK1 (0.41) JAK2
SCHEMBL24865487 0.81 TTK (0.34) SYKHTR1AHTR2ADCLK1LRRK2
SCHEMBL30336110 0.80 ROCK2 (0.47) JAK2LRRK2
SCHEMBL24865568 0.80 ROCK2 (0.47) JAK2LRRK2
SCHEMBL24865403 0.80 TTK (0.39) DCLK1LRRK2
SCHEMBL24864899 0.79 ADRB1 (0.33) BCL6DCLK1LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117999259-A Iron death modulators, their preparation and use 维泰瑞隆有限公司 2024-05-07 CN disclosed
WO-2023280296-A1 FERROPTOSIS MODULATORS, PREPARATIONS, AND USES THEREOF Sironax Ltd. (KY) 2023-01-12 WO disclosed