SCHEMBL24865673

SCHEMBL24865673

O=c1[nH]c2cc(Nc3ccc(N4CCC(C(F)(F)F)CC4)cc3)ccc2o1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 7/20 0.41
JAK3 P52333 7/20 0.41
CNR2 P34972 1/20 0.39
JAK2 O60674 3/20 0.39
CYP3A4 P08684 3/20 0.39
SYK P43405 1/20 0.38
P2RX3 P56373 1/20 0.38
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31123276 1.00 JAK1 (0.41) JAK1JAK3CNR2JAK2CYP3A4
SCHEMBL24865172 0.87 JAK1 (0.41) JAK1JAK3JAK2CYP3A4P2RX3
SCHEMBL31123300 0.87 JAK1 (0.41) JAK1JAK3JAK2CYP3A4P2RX3
SCHEMBL24864995 0.79 ACHE (0.46) CNR2
SCHEMBL31123262 0.79 MEN1 (0.39)
SCHEMBL24865555 0.79 MEN1 (0.39)
SCHEMBL31123319 0.77 BCL6 (0.40) JAK1JAK3CNR2SYK
SCHEMBL24865678 0.77 BCL6 (0.40) JAK1JAK3CNR2SYK
SCHEMBL24865740 0.77 BCL6 (0.40) JAK1JAK3CNR2
SCHEMBL24865697 0.76 MAPT (0.45) JAK1JAK3JAK2CYP3A4SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117999259-A Iron death modulators, their preparation and use 维泰瑞隆有限公司 2024-05-07 CN disclosed
WO-2023280296-A1 FERROPTOSIS MODULATORS, PREPARATIONS, AND USES THEREOF Sironax Ltd. (KY) 2023-01-12 WO disclosed