SCHEMBL24865348

SCHEMBL24865348

CNCCN1C(=O)COc2cc(Nc3ccc(C(C)(C)C)cc3)ccc21

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.41
PIK3CG P48736 2/20 0.39
CHRM5 P08912 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
EGFR P00533 2/20 0.36
RORC P51449 1/20 0.35
MAPT P10636 1/20 0.35
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30336656 1.00 ALDH1A1 (0.44) ALDH1A1POLBPIK3CGCHRM5CHRM1
SCHEMBL24864939 0.88 ALDH1A1 (0.47) ALDH1A1POLBPIK3CGCHRM5CHRM1
SCHEMBL30336220 0.88 ALDH1A1 (0.47) ALDH1A1POLBPIK3CGCHRM5CHRM1
SCHEMBL29209064 0.85 ALDH1A1 (0.46) ALDH1A1POLBPIK3CGL3MBTL1RORC
SCHEMBL24865349 0.83 GABRG2 (0.46) ALDH1A1POLBGABRG2GABRB3GABRA5
SCHEMBL30336271 0.83 GABRG2 (0.46) ALDH1A1POLBGABRG2GABRB3GABRA5
SCHEMBL24865351 0.80 MAPT (0.41) CHRM5CHRM1CHRM3GABRG2GABRB3
SCHEMBL30336252 0.80 GABRG2 (0.35) POLBCHRM5CHRM1CHRM3GABRG2
SCHEMBL24865447 0.80 GABRG2 (0.35) POLBCHRM5CHRM1CHRM3GABRG2
SCHEMBL31123245 0.79 ALDH1A1 (0.42) ALDH1A1POLBPIK3CGL3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117999259-A Iron death modulators, their preparation and use 维泰瑞隆有限公司 2024-05-07 CN disclosed
WO-2023280296-A1 FERROPTOSIS MODULATORS, PREPARATIONS, AND USES THEREOF Sironax Ltd. (KY) 2023-01-12 WO disclosed