SCHEMBL24865447

SCHEMBL24865447

CNCCN1C(=O)COc2cc(Nc3ccc(C4CC(C)OC(C)C4)cc3)ccc21

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
SCD O00767 1/20 0.34
EGFR P00533 5/20 0.33
RORC P51449 1/20 0.33
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33
POLB P06746 1/20 0.32
TSHR P16473 1/20 0.32
PLK1 P53350 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30336252 1.00 GABRG2 (0.35) GABRG2GABRB3GABRA5CHRM5CHRM1
SCHEMBL24864971 0.85 GABRA5 (0.44) GABRG2GABRB3GABRA5
SCHEMBL30336693 0.85 GABRA5 (0.44) GABRG2GABRB3GABRA5
SCHEMBL24865351 0.85 MAPT (0.41) GABRG2GABRB3GABRA5CHRM5CHRM1
SCHEMBL30336550 0.82 BRD4 (0.35) GABRG2GABRB3GABRA5CHRM5CHRM1
SCHEMBL24864948 0.82 BRD4 (0.35) GABRG2GABRB3GABRA5CHRM5CHRM1
SCHEMBL30336656 0.80 ALDH1A1 (0.44) GABRG2GABRB3GABRA5CHRM5CHRM1
SCHEMBL24865348 0.80 ALDH1A1 (0.44) GABRG2GABRB3GABRA5CHRM5CHRM1
SCHEMBL24865445 0.80 NOS3 (0.34) CHRM5CHRM1CHRM3RORCITGB3
SCHEMBL24865328 0.79 EGFR (0.37) CHRM5CHRM1CHRM3EGFRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117999259-A Iron death modulators, their preparation and use 维泰瑞隆有限公司 2024-05-07 CN disclosed
WO-2023280296-A1 FERROPTOSIS MODULATORS, PREPARATIONS, AND USES THEREOF Sironax Ltd. (KY) 2023-01-12 WO disclosed