SCHEMBL24865620

SCHEMBL24865620

CNc1ccc(Nc2ccc(N3CCC(C(F)(F)F)CC3)cc2)cc1C#N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38
KCNH2 Q12809 1/20 0.38
CCNT1 O60563 2/20 0.36
CDK1 P06493 2/20 0.36
CCNB1 P14635 2/20 0.36
CCNA2 P20248 2/20 0.36
CDK2 P24941 2/20 0.36
CDK7 P50613 2/20 0.36
CDK9 P50750 2/20 0.36
CCNH P51946 2/20 0.36
PIK3CD O00329 1/20 0.36
PRKAB2 O43741 1/20 0.36
NUAK1 O60285 1/20 0.36
ABL1 P00519 1/20 0.36
FYN P06241 1/20 0.36
CSF1R P07333 1/20 0.36
RET P07949 1/20 0.36
PDGFRB P09619 1/20 0.36
FGFR1 P11362 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30336093 1.00 DRD2 (0.38) DRD2DRD3KCNH2CCNT1CDK1
SCHEMBL31053582 0.83 IDO1 (0.44) DRD2DRD3KCNH2JAK2TBK1
SCHEMBL25193116 0.82 AR (0.47) DRD2DRD3KCNH2MAPTAR
SCHEMBL24865618 0.80 CNR2 (0.36) JAK2MEN1ALDH1A1MAPTKMT2A
SCHEMBL30885112 0.80 CNR2 (0.36) JAK2MEN1ALDH1A1MAPTKMT2A
SCHEMBL1664150 0.78 SMN1; SMN2 (0.41) ABL1JAK2TBK1MEN1ALDH1A1
SCHEMBL25042072 0.78 HRH3 (0.47) MEN1ALDH1A1MAPTKMT2AKDM4E
SCHEMBL31053626 0.76 CCNA2 (0.41) DRD2DRD3KCNH2CCNA2CDK2
SCHEMBL25193652 0.76 CCNA2 (0.41) DRD2DRD3KCNH2CCNA2CDK2
SCHEMBL24865745 0.76 MAPK10 (0.44) FGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117999259-A Iron death modulators, their preparation and use 维泰瑞隆有限公司 2024-05-07 CN disclosed
WO-2023280296-A1 FERROPTOSIS MODULATORS, PREPARATIONS, AND USES THEREOF Sironax Ltd. (KY) 2023-01-12 WO disclosed