SCHEMBL24865757

SCHEMBL24865757

Cn1c(=O)oc2cc(Nc3ccc(N4CCC(O)(C(F)(F)F)CC4)cc3)ccc21

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
ALDH1A1 P00352 2/20 0.41
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA5 P31644 1/20 0.40
PKM P14618 1/20 0.39
GFER P55789 1/20 0.39
LMNA P02545 2/20 0.39
MAPT P10636 2/20 0.39
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 2/20 0.38
HTR1A P08908 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31123282 1.00 KDM4E (0.43) KDM4EMEN1KMT2AALDH1A1GABRG2
SCHEMBL24865793 0.86 ALDH1A1 (0.41) KDM4EMEN1KMT2AALDH1A1GABRG2
SCHEMBL31123224 0.83 SMN1; SMN2 (0.47) ALDH1A1PKMLMNASMN1; SMN2TP53
SCHEMBL24865602 0.83 SMN1; SMN2 (0.47) ALDH1A1PKMLMNASMN1; SMN2TP53
SCHEMBL24865639 0.81 GABRG2 (0.43) KDM4EMEN1KMT2AALDH1A1GABRG2
SCHEMBL31123316 0.81 GABRG2 (0.46) KDM4EMEN1KMT2AALDH1A1GABRG2
SCHEMBL24865238 0.81 GABRG2 (0.46) KDM4EMEN1KMT2AALDH1A1GABRG2
SCHEMBL30336455 0.78 KDM4E (0.47) KDM4EMEN1KMT2AALDH1A1GABRG2
SCHEMBL24865120 0.78 KDM4E (0.47) KDM4EMEN1KMT2AALDH1A1GABRG2
SCHEMBL24865689 0.78 ALDH1A1 (0.35) MEN1KMT2AALDH1A1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117999259-A Iron death modulators, their preparation and use 维泰瑞隆有限公司 2024-05-07 CN disclosed
WO-2023280296-A1 FERROPTOSIS MODULATORS, PREPARATIONS, AND USES THEREOF Sironax Ltd. (KY) 2023-01-12 WO disclosed