SCHEMBL2487494

SCHEMBL2487494

O=C(O)Oc1cn(Cc2ccc(-c3ccncc3F)cc2F)c2c(F)ccc(F)c2c1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 9/20 0.40
RIPK3 Q9Y572 1/20 0.35
METAP2 P50579 1/20 0.34
BDKRB1 P46663 2/20 0.33
MAP4K4 O95819 2/20 0.33
PRKACA P17612 2/20 0.33
CDK2 P24941 2/20 0.33
GSK3B P49841 2/20 0.33
CLK4 Q9HAZ1 2/20 0.33
CDC7 O00311 1/20 0.33
ROCK2 O75116 1/20 0.33
HIPK2 Q9H2X6 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
CTSA P10619 2/20 0.32
ICMT O60725 1/20 0.32
SLC22A12 Q96S37 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.31
PRKCG P05129 1/20 0.31
CDK1 P06493 1/20 0.31
RPS6KB1 P23443 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2487909 0.87 CHRM1 (0.43) CHRM1
SCHEMBL2492208 0.86 CHRM1 (0.41) CHRM1PTGDR2
SCHEMBL2487841 0.86 CHRM1 (0.55) CHRM1RIPK3METAP2MAP4K4PRKACA
SCHEMBL2486084 0.84 CHRM1 (0.53) CHRM1BDKRB1PTGDR2
SCHEMBL2492205 0.83 CHRM1 (0.41) CHRM1ROCK2PTGDR2
SCHEMBL2488348 0.83 CHRM1 (0.40) CHRM1
SCHEMBL2487937 0.83 CHRM1 (0.42) CHRM1METAP2MAP4K4PRKACACDK2
SCHEMBL2488465 0.82 CHRM1 (0.41) CHRM1PTGDR2
SCHEMBL2487485 0.81 CHRM1 (0.45) CHRM1METAP2
SCHEMBL2491881 0.80 ERN1 (0.42) CHRM1RPS6KA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2037739-B1 BENZYL-SUBSTITUTED QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK SHARP & DOHME (US) 2011-10-26 EP claimed