SCHEMBL24876264

SCHEMBL24876264

COc1ccc(-c2ccc(NS(=O)(=O)c3cc(N)c(N)cc3C)cc2Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.50
ALDH1A1 P00352 4/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
HPGD P15428 2/20 0.50
THRB P10828 3/20 0.47
IDH1 O75874 1/20 0.47
PLAU P00749 1/20 0.46
PKM P14618 1/20 0.45
BRD4 O60885 1/20 0.45
BRD2 P25440 1/20 0.45
BRD3 Q15059 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CDK1 P06493 1/20 0.44
CCNB1 P14635 1/20 0.44
CCNA2 P20248 1/20 0.44
CDK2 P24941 1/20 0.44
CDK7 P50613 1/20 0.44
CCNH P51946 1/20 0.44
CCNA1 P78396 1/20 0.44
FFAR4 Q5NUL3 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24876266 0.84 CDK1 (0.48) LMNAALDH1A1SMN1; SMN2HPGDTHRB
SCHEMBL31679961 0.83 THRB (0.70) LMNAALDH1A1SMN1; SMN2HPGDTHRB
SCHEMBL24876270 0.79 TSHR (0.48) LMNAALDH1A1SMN1; SMN2HPGDIDH1
SCHEMBL24876629 0.78 HSD17B2 (0.43) LMNATHRBIDH1PKMCDK1
SCHEMBL3376228 0.78 EPHX2 (0.55) LMNAHPGDPLAUCYP19A1TP53
SCHEMBL24876762 0.78 LMNA (0.44) LMNATHRBPKMCDK1CCNB1
SCHEMBL31679941 0.77 THRB (0.64) LMNAALDH1A1SMN1; SMN2HPGDTHRB
SCHEMBL10576667 0.75 ALDH1A1 (0.55) LMNAALDH1A1SMN1; SMN2HPGDTHRB
SCHEMBL24876673 0.74 THRB (0.70) LMNATHRBIDH1PKMMAPT
SCHEMBL24876669 0.74 LMNA (0.43) LMNAALDH1A1SMN1; SMN2HPGDTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023280970-A1 INHIBITORS OF ALPHA-HEMOLYSIN OF STAPHYLOCOCCUS AUREUS Helmholtz-Zentrum für Infektionsforschung GmbH (DE) 2023-01-12 WO disclosed