SCHEMBL2488050

SCHEMBL2488050

FC(F)(F)c1ccccc1-c1ncc2nc[nH]c2n1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 9/20 0.48
CYP2C19 P33261 7/20 0.48
CYP3A4 P08684 6/20 0.48
ALDH1A1 P00352 1/20 0.48
USP1 O94782 10/20 0.47
WDR48 Q8TAF3 10/20 0.47
TSHR P16473 3/20 0.45
HSD17B10 Q99714 3/20 0.45
ALOX15 P16050 1/20 0.45
MAPK1 P28482 1/20 0.45
HIF1A Q16665 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
CYP2D6 P10635 5/20 0.43
CYP2C9 P11712 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
RECQL P46063 2/20 0.43
CLK4 Q9HAZ1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6944922 0.78 CYP1A2 (0.45) CYP1A2CYP2C19CYP3A4ALDH1A1TSHR
SCHEMBL29240141 0.77 GSK3B (0.41) CYP1A2CYP3A4ALDH1A1TSHRHSD17B10
SCHEMBL30630379 0.74 TRPA1 (0.38) CYP1A2CYP2C19CYP3A4ALDH1A1HSD17B10
SCHEMBL8390254 0.74 USP1 (0.55) CYP1A2CYP2C19CYP3A4ALDH1A1USP1
SCHEMBL4156258 0.74 USP1 (0.52) CYP1A2CYP2C19CYP3A4ALDH1A1USP1
SCHEMBL10783430 0.74 CYP1A2 (0.50) CYP1A2CYP2C19CYP3A4ALDH1A1USP1
SCHEMBL680853 0.73 NPC1 (0.45) CYP3A4ALDH1A1HSD17B10MAPK1MEN1
Hydrochloric Acid SCHEMBL4456673 0.72 NPC1 (0.44) CYP3A4ALDH1A1HSD17B10MAPK1MEN1
SCHEMBL30707907 0.70 USP1 (0.39) USP1
SCHEMBL4924089 0.70 KDM4E (0.48) CYP1A2HSD17B10ALOX15MAPK1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379555-A1 PURINE COMPOUNDS Eli Lilly and Company (US) 2011-10-26 EP claimed
WO-2010080306-A1 PURINE COMPOUNDS ELI LILLY AND COMPANY (US) 2010-07-15 WO claimed