SCHEMBL6944922

SCHEMBL6944922

Cc1ccccc1-c1ncc2nc[nH]c2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 12/20 0.45
CYP3A4 P08684 9/20 0.45
CYP2C19 P33261 8/20 0.45
CYP2D6 P10635 8/20 0.40
HSD17B10 Q99714 7/20 0.40
CLK4 Q9HAZ1 5/20 0.40
ALOX15 P16050 3/20 0.40
USP2 O75604 2/20 0.40
CYP2C9 P11712 1/20 0.40
GAA P10253 3/20 0.39
IDO1 P14902 1/20 0.39
METAP2 P50579 1/20 0.39
ALDH1A1 P00352 7/20 0.39
TSHR P16473 3/20 0.39
MAPK1 P28482 3/20 0.39
DCUN1D1 Q96GG9 1/20 0.38
HIF1A Q16665 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29240141 0.80 GSK3B (0.41) CYP1A2CYP3A4HSD17B10ALOX15GAA
SCHEMBL2488050 0.78 CYP1A2 (0.48) CYP1A2CYP3A4CYP2C19CYP2D6HSD17B10
SCHEMBL30630379 0.78 TRPA1 (0.38) CYP1A2CYP3A4CYP2C19CYP2D6HSD17B10
SCHEMBL30850611 0.77 BRAF (0.42) HSD17B10GAAALDH1A1HPGDKDM4E
SCHEMBL680853 0.77 NPC1 (0.45) CYP3A4HSD17B10GAAALDH1A1MAPK1
SCHEMBL30707907 0.77 USP1 (0.39)
SCHEMBL27436087 0.76 ALOX5AP (0.46) CYP1A2CYP3A4CYP2C19CYP2D6HSD17B10
SCHEMBL18725509 0.76 PDK2 (0.31) HSD17B10GAAALDH1A1HPGDKDM4E
Hydrochloric Acid SCHEMBL4456673 0.76 NPC1 (0.44) CYP3A4HSD17B10GAAALDH1A1MAPK1
SCHEMBL4924089 0.73 KDM4E (0.48) CYP1A2HSD17B10ALOX15METAP2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed