SCHEMBL2488055

SCHEMBL2488055

FC(F)(F)c1ccccc1-c1nc2cncnc2[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 13/20 0.50
CYP2C19 P33261 12/20 0.50
CYP2D6 P10635 11/20 0.50
ALDH1A1 P00352 7/20 0.50
ALOX15 P16050 6/20 0.50
HSD17B10 Q99714 6/20 0.50
MAPK1 P28482 2/20 0.50
CYP1A2 P05177 10/20 0.48
TDP1 Q9NUW8 4/20 0.48
HDAC3 O15379 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
PTGES O14684 1/20 0.46
USP2 O75604 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
PARP1 P09874 1/20 0.43
NPY5R Q15761 1/20 0.43
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3063543 0.81 NPC1 (0.54) ALDH1A1HSD17B10PTGESPARP1KDM4E
SCHEMBL6944926 0.78 ALDH1A1 (0.54) CYP3A4CYP2C19CYP2D6ALDH1A1ALOX15
SCHEMBL3058557 0.76 NPC1 (0.41) ALDH1A1PTGES
SCHEMBL28024969 0.74 NPBWR1 (0.49)
SCHEMBL30874472 0.74 MKNK1 (0.58) ALDH1A1HSD17B10MEN1KMT2AKDM4E
SCHEMBL5914424 0.74 KDM4C (0.49) CYP3A4ALDH1A1ALOX15HSD17B10MAPK1
SCHEMBL10740426 0.74 HDAC3 (0.53) ALDH1A1HSD17B10HDAC3HDAC7HDAC10
SCHEMBL5240824 0.73 NPC1 (0.41) CYP2D6ALDH1A1MAPK1MEN1KMT2A
SCHEMBL4117692 0.73 NPC1 (0.63) ALDH1A1HSD17B10MAPK1HDAC3HDAC7
SCHEMBL31679092 0.73 NPC1 (0.63) ALDH1A1HSD17B10MAPK1HDAC3HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379555-A1 PURINE COMPOUNDS Eli Lilly and Company (US) 2011-10-26 EP claimed
WO-2010080306-A1 PURINE COMPOUNDS ELI LILLY AND COMPANY (US) 2010-07-15 WO claimed