SCHEMBL2489241

SCHEMBL2489241

OB(OOCc1ccccc1)c1cnc(Cl)nc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.38
LIPE Q05469 1/20 0.37
POLB P06746 1/20 0.35
PLAU P00749 1/20 0.35
ALDH1A1 P00352 2/20 0.34
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
PTGS1 P23219 1/20 0.34
SLC6A2 P23975 1/20 0.34
CYP2C19 P33261 1/20 0.34
PTGS2 P35354 1/20 0.34
SLC6A3 Q01959 1/20 0.34
HIF1A Q16665 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
P4HTM Q9NXG6 1/20 0.34
TSHR P16473 1/20 0.33
P2RX7 Q99572 1/20 0.33
LTA4H P09960 1/20 0.33
MAPK14 Q16539 1/20 0.33
ALKBH1 Q13686 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3714673 0.80 TSHR (0.43) LIPEALDH1A1LMNACYP1A2PTGS1
SCHEMBL18586876 0.76 ORAI1 (0.47) POLBALDH1A1CYP1A2CYP2C19IDO1
SCHEMBL28857039 0.76 KMT2A (0.46) POLBALDH1A1LMNACYP1A2CYP2C19
SCHEMBL3658498 0.73 IDO1 (0.40) LIPELMNAIDO1ENPP2
SCHEMBL28652344 0.70 TSHR (0.48) LIPEALDH1A1LMNACYP1A2PTGS1
SCHEMBL18586469 0.70 IDO1 (0.40) LIPEALDH1A1LMNAIDO1
SCHEMBL18587306 0.70 NPC1 (0.42) LIPEPOLBLMNA
SCHEMBL17674482 0.70 KMT2A (0.44) PIN1POLBALDH1A1LMNASLC6A2
SCHEMBL457443 0.70 P4HTM (0.53) PIN1LMNACYP1A2PTGS1SLC6A2
SCHEMBL3723968 0.68 ENPP2 (0.53) CYP1A2LTA4HIDO1ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379534-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2011-10-26 EP disclosed
WO-2010072598-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-07-01 WO disclosed