SCHEMBL28857039

SCHEMBL28857039

OB(OOCc1ccccc1)c1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.46
LMNA P02545 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
CYP19A1 P11511 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
NAPRT Q6XQN6 1/20 0.39
MAPK1 P28482 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HIF1A Q16665 1/20 0.39
KCNA5 P22460 1/20 0.39
MEN1 O00255 1/20 0.39
RAB9A P51151 1/20 0.38
SGMS2 Q8NHU3 1/20 0.38
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3714673 0.84 TSHR (0.43) KMT2ALMNATDP1MAPK1CYP1A2
SCHEMBL26985702 0.80 LMNA (0.36) KMT2ALMNATDP1CYP19A1CYP11B1
SCHEMBL3658498 0.76 IDO1 (0.40) LMNA
SCHEMBL2489241 0.76 PIN1 (0.38) LMNACYP1A2CYP2C19HIF1AALDH1A1
SCHEMBL568870 0.74 ALDH1A1 (0.41) KMT2ALMNANAPRTCYP1A2CYP3A4
SCHEMBL18586876 0.73 ORAI1 (0.47) KMT2ATDP1CYP1A2CYP3A4CYP2C9
SCHEMBL18586469 0.73 IDO1 (0.40) KMT2ALMNAMEN1RAB9AALDH1A1
SCHEMBL18587306 0.73 NPC1 (0.42) LMNATDP1RAB9APOLB
SCHEMBL8131766 0.73 ALDH1A1 (0.41) KMT2ALMNATDP1NAPRTCYP1A2
SCHEMBL13712395 0.71 F7 (0.39) KMT2ALMNATDP1NAPRTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117916231-A Compounds for inhibiting or degrading target proteins, compositions comprising the same, methods of making and methods of using the same 纽力克斯治疗公司 2024-04-19 CN disclosed
CN-117813307-A Difunctional degradants of interleukin-1 receptor related kinase and therapeutic uses thereof 新锐思生物制药股份有限公司 2024-04-02 CN disclosed
CN-117693502-A Compounds for inhibiting or degrading ITK, compositions comprising the same, methods of making the same, and methods of using the same 纽力克斯治疗公司 2024-03-12 CN disclosed
CN-115003304-A Bifunctional compounds for the degradation of BTK via the ubiquitin proteasome pathway 纽力克斯治疗公司 2022-09-02 CN disclosed