SCHEMBL24897752

SCHEMBL24897752

O=C1Nc2cc(F)c(F)cc2C1(F)F

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.36
PGR P06401 1/20 0.33
CYP1A2 P05177 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
MDM2 Q00987 1/20 0.31
POLB P06746 1/20 0.31
CASP6 P55212 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31677515 0.84 IDO1 (0.39) IDO1PGR
SCHEMBL7825677 0.77 PGR (0.50) PGR
SCHEMBL2827536 0.75 CYP1A2 (0.57) IDO1PGRCYP1A2MAPTCYP2C19
SCHEMBL29860253 0.75 PGR (0.44) PGRCYP1A2MAPTCYP2C19
SCHEMBL24898308 0.72 POLB (0.34) IDO1PGRPOLBCASP6
SCHEMBL30211424 0.72 POLB (0.34) IDO1PGRPOLBCASP6
SCHEMBL24898318 0.71 PKM (0.35)
SCHEMBL17950681 0.71 KMT2A (0.66) PGRCYP1A2MAPTCYP2C19KMT2A
SCHEMBL25115048 0.69 IDO1 (0.43) IDO1PGRCYP1A2MAPTCYP2C19
SCHEMBL30548920 0.69 IDO1 (0.43) IDO1CYP1A2MAPTCYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023288242-A1 PI3Kα INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2023-01-19 WO disclosed
CN-108299137-B Selective fluorination method of isatin hydrazone compound 中南大学 2020-04-14 CN disclosed