SCHEMBL2489944

SCHEMBL2489944

COc1ccc(Cn2ncc3c4c(cnc32)CN(C(Cl)(C=O)c2ccccc2)CC4)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.42
MAPT P10636 5/20 0.42
LMNA P02545 3/20 0.42
ALOX15 P16050 2/20 0.42
HPGD P15428 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HSD17B10 Q99714 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.38
NPBWR1 P48145 4/20 0.37
ADORA1 P30542 3/20 0.37
CNR2 P34972 2/20 0.36
PKM P14618 2/20 0.36
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
POLB P06746 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPK1 P28482 1/20 0.35
NTSR1 P30989 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2489975 0.80 ALDH1A1 (0.43) ALDH1A1MAPTLMNAALOX15HPGD
SCHEMBL2489846 0.79 ABCB1 (0.47) ALDH1A1MAPTLMNAALOX15HPGD
SCHEMBL12315714 0.79 ALDH1A1 (0.48) ALDH1A1MAPTLMNAALOX15HPGD
SCHEMBL2487710 0.78 LMNA (0.45) ALDH1A1MAPTLMNAALOX15HPGD
SCHEMBL2488683 0.78 FAAH (0.52) ALDH1A1MAPTLMNAALOX15HPGD
SCHEMBL2489970 0.78 KMT2A (0.48) ALDH1A1MAPTLMNAALOX15HPGD
SCHEMBL2485333 0.77 HPGD (0.52) ALDH1A1MAPTLMNAALOX15HPGD
SCHEMBL2488514 0.77 ADORA1 (0.46) ALDH1A1MAPTLMNAALOX15HPGD
SCHEMBL2488863 0.77 ALDH1A1 (0.43) ALDH1A1MAPTLMNAALOX15HPGD
SCHEMBL2802729 0.76 ALDH1A1 (0.38) ALDH1A1MAPTLMNAALOX15HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379551-A1 SUBSTITUTED PYRAZOLO [3, 4-B]PYRIDINE COMPOUNDS ArQule, Inc. (US) 2011-10-26 EP disclosed
WO-2010078427-A1 SUBSTITUTED PYRAZOLO [3, 4-B] PYRIDINE COMPOUNDS ARQULE, INC. (US) 2010-07-08 WO disclosed