SCHEMBL24900076

SCHEMBL24900076

CCCc1cc(N)nc2c1c(C)nn2C

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 2/20 0.47
NOS2 P35228 2/20 0.39
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
PDE5A O76074 8/20 0.38
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 3/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 2/20 0.36
GAA P10253 1/20 0.35
MAPK1 P28482 1/20 0.35
CLK1 P49759 1/20 0.35
UBE2N P61088 1/20 0.35
IKBKB O14920 1/20 0.34
BCDIN3D Q7Z5W3 1/20 0.32
PDE10A Q9Y233 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12073695 0.72 S1PR2 (0.46) S1PR2NOS2NOS3NOS1KDM4E
SCHEMBL18314725 0.70 NOS2 (0.48) NOS2NOS3NOS1IKBKB
SCHEMBL18310645 0.65 NOS2 (0.43) NOS2NOS3NOS1KDM4EALDH1A1
SCHEMBL18310670 0.65 NOS2 (0.43) NOS2NOS3NOS1IKBKB
SCHEMBL21183232 0.64 DYRK1A (0.38) PDE5AKDM4EALDH1A1GAABCDIN3D
SCHEMBL4841951 0.64 DHFR (0.36) KDM4EALDH1A1GAABCDIN3DPDE10A
SCHEMBL423531 0.63 MEN1 (0.60) S1PR2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL17229299 0.62 NOS2 (0.44) NOS2NOS3NOS1KDM4EALDH1A1
SCHEMBL8142879 0.62 HRH4 (0.37) PDE5AKDM4EALDH1A1HPGDHSD17B10
SCHEMBL23369560 0.62 ADORA2A (0.40) NOS2NOS3NOS1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023283921-A1 DPD INHIBITOR, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF 北京深蓝泰医药科技有限公司 2023-01-19 WO disclosed