SCHEMBL2490671

SCHEMBL2490671

NC(=O)N(c1cccnc1Cl)C1CCN(OC(=O)OCc2ccccc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.38
CYP2C19 P33261 1/20 0.38
GRIN2B Q13224 2/20 0.37
OPRM1 P35372 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CHRM2 P08172 1/20 0.35
CHRM3 P20309 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
ENPP2 Q13822 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1285381 0.87 SMN1; SMN2 (0.54) POLBSMN1; SMN2CYP2C19GRIN2BNPC1
SCHEMBL30006056 0.82 CHRM3 (0.53) OPRM1CHRM2CHRM3
SCHEMBL27092754 0.82 CHRM3 (0.53) OPRM1CHRM2CHRM3
SCHEMBL3063074 0.77 RPLP1 (0.38) SMN1; SMN2CYP2C19CHRM2CHRM3
SCHEMBL2492658 0.77 POLB (0.46) POLBSMN1; SMN2GRIN2BL3MBTL1NPC1
SCHEMBL3064320 0.76 CYP2C19 (0.50) SMN1; SMN2CYP2C19GRIN2BL3MBTL1CHRM2
SCHEMBL4762750 0.75 ALDH1A1 (0.43) SMN1; SMN2CYP2C19OPRM1
SCHEMBL19873844 0.75 OPRD1 (0.43) OPRM1
SCHEMBL4564976 0.74 SLC6A15 (0.44) POLBSMN1; SMN2CYP2C19GRIN2BL3MBTL1
SCHEMBL27769658 0.72 ALDH1A1 (0.39) OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225223-B1 ORGANIC COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2017-01-11 EP disclosed
EP-2225236-B1 ORGANIC COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2016-01-27 EP disclosed
EP-2379529-B1 CGRP-ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2015-06-10 EP disclosed
EP-2205590-B1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2014-06-04 EP disclosed
EP-2379529-A1 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-10-26 EP disclosed
EP-2251338-A2 Organic compounds Boehringer Ingelheim International GmbH (DE) 2010-11-17 EP disclosed
EP-2225223-A2 ORGANIC COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2010-09-08 EP disclosed
EP-2225236-A2 ORGANIC COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2010-09-08 EP disclosed
EP-2205590-A1 CGRP ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2010-07-14 EP disclosed
WO-2010070022-A1 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-06-24 WO disclosed
WO-2010020628-A1 NOVEL PRODUCTION METHOD FOR L-PIPERIDINE-4-YL-1,3-DIHYDRO-IMIDAZO [4,5-B] PYRIDINE-2-ONE AND MONO- AND DIHYDROCHLORIDES THEREOF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-02-25 WO disclosed
WO-2009065921-A2 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-05-28 WO disclosed
WO-2009065919-A2 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-05-28 WO disclosed
WO-2009050235-A1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-04-23 WO disclosed
WO-2009050232-A1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-04-23 WO disclosed