SCHEMBL2490883

SCHEMBL2490883

O=[C]c1cc(I)ccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
IDO1 P14902 1/20 0.33
VCAM1 P19320 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21201454 0.82 IDO1 (0.37) MAPK1TDP1IDO1
SCHEMBL3336251 0.77 VCAM1 (0.48) MAPK1IDO1VCAM1
SCHEMBL95478 0.76 TP53 (0.48) MAPK1TDP1VCAM1
SCHEMBL6212276 0.73 PTGDR2 (0.36) MAPK1TDP1VCAM1
SCHEMBL6897410 0.73 ALDH1A1 (0.40) MAPK1TDP1VCAM1
SCHEMBL95554 0.71 ERN1 (0.31)
SCHEMBL80565 0.69
SCHEMBL30469268 0.69
SCHEMBL2515789 0.68 PTGDR2 (0.43)
SCHEMBL5969859 0.68 ACACB (0.42) MAPK1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111410639-B Preparation method of empagliflozin intermediate impurity 天津法莫西医药科技有限公司 2021-02-26 CN disclosed
CN-111410639-A Preparation method of empagliflozin intermediate impurity 天津法莫西医药科技有限公司 2020-07-14 CN disclosed
EP-2183263-B1 METHODS AND COMPOUNDS USEFUL FOR THE PREPARATION OF SODIUM GLUCOSE CO-TRANSPORTER 2 INHIBITORS LEXICON PHARMACEUTICALS INC (US) 2011-10-26 EP disclosed
CN-1161336-C Quinoline carboxamides as antiviral agents �������Ŷ���Լ��������˾ 2004-08-11 CN disclosed
CN-1333753-A Quinoline carboxamides as antiviral agents UPJOHN CO (US) 2002-01-30 CN disclosed