Piperidolate

Piperidolate

SCHEMBL249131

CCN1CCCC(OC(=O)C(c2ccccc2)c2ccccc2)C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 1.00
CYP3A4 P08684 3/20 1.00
CYP1A2 P05177 3/20 1.00
HTT P42858 1/20 0.71
TP53 P04637 1/20 0.56
PKM P14618 1/20 0.56
NFKB1 P19838 1/20 0.56
THPO P40225 1/20 0.56
HIF1A Q16665 1/20 0.56
KDM4E B2RXH2 1/20 0.56
LMNA P02545 3/20 0.55
THRB P10828 3/20 0.55
BLM P54132 3/20 0.55
PMP22 Q01453 3/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
GMNN O75496 1/20 0.55
ALDH1A1 P00352 1/20 0.55
MAPT P10636 1/20 0.55
CHRM2 P08172 5/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Piperidolate SCHEMBL28832658 1.00 CYP2D6 (1.00) CYP2D6CYP3A4CYP1A2HTTTP53
Piperidolate SCHEMBL437741 0.99 CYP3A4 (1.00) CYP2D6CYP3A4CYP1A2HTTTP53
Piperidolate SCHEMBL2734595 0.99 CYP2D6 (0.98) CYP2D6CYP3A4CYP1A2HTTTP53
Piperidolate SCHEMBL1649482 0.98 CYP2D6 (0.95) CYP2D6CYP3A4CYP1A2HTTTP53
SCHEMBL14128808 0.92 CYP2D6 (0.86) CYP2D6CYP3A4CYP1A2HTTTP53
SCHEMBL14125434 0.92 CYP2D6 (0.86) CYP2D6CYP3A4CYP1A2HTTTP53
SCHEMBL24671287 0.86 CYP3A4 (0.76) CYP2D6CYP3A4CYP1A2HTTTP53
SCHEMBL7588607 0.84 CYP2D6 (0.73) CYP2D6CYP3A4CYP1A2HTTTP53
SCHEMBL24671171 0.83 CYP2D6 (1.00) CYP2D6CYP3A4CYP1A2HTTTP53
SCHEMBL10517675 0.80 CYP2D6 (0.70) CYP2D6CYP3A4CYP1A2HTTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 475 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026100654-A1 NUCLEIC ACID INTRODUCTION AID, NUCLEIC ACID INTRODUCTION AGENT, AND NUCLEIC ACID INTRODUCTION METHOD 株式会社インファーマシア 2026-05-15 WO claimed
EP-4154879-B1 PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING NICOTINE WITHDRAWAL SYMPTOMS KOREA INST SCI & TECH (KR) 2025-09-10 EP claimed
WO-2025038382-A1 PHARMACEUTICAL ADHESIVE COMPOSITIONS MOMENTIVE PERFORMANCE MATERIALS INC. (US) 2025-02-20 WO claimed
EP-4154879-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING NICOTINE WITHDRAWAL SYMPTOMS Korea Institute of Science and Technology (KR) 2023-03-29 EP claimed
US-11065205-B2 Immediate/delayed drug delivery DRUG DELIVERY INTERNATIONAL LIMITED (GB) 2021-07-20 US claimed
US-20210154208-A1 Method to Identify Agents That Can Overcome Inhibition Caused By Drug-protein Binding of the Human Plasma Protein, Alpha-1-acid Glycoprotein THE JOHNS HOPKINS UNIVERSITY 2021-05-27 US claimed
US-10987316-B2 Compositions and methods for transdermal delivery of tertiary amine drugs NOVEN PHARMACEUTICALS, INC. (US) 2021-04-27 US claimed
EP-3773556-A1 COMPOSITIONS AND METHODS FOR INCREASING REMYELINATION Frequency Therapeutics, Inc. (US) 2021-02-17 EP claimed
US-10689370-B2 Cyclopropane carboxamide modulators of cystic fibrosis transmembrane conductance regulator AUSPEX PHARMACEUTICALS, INC. (US) 2020-06-23 US claimed
US-20190336490-A1 COMPOSITIONS AND METHODS FOR INCREASING REMYELINATION Frequency Therapeutics, Inc. 2019-11-07 US claimed
EP-2026807-A1 USE OF PARASYMPATHOLYTIC SUBSTANCES TO ENHANCE AND ACCELERATE STEM CELL DIFFERENTIATION, RELATED METHOD AND COMPOSITIONS Universita' Degli Studi di Torino (IT) 2009-02-25 EP claimed
WO-2009018169-A1 SUBSTITUTED CYCLOHEXANOLS AUSPEX PHARMACEUTICALS, INC. (US) 2009-02-05 WO claimed
US-20090028873-A1 SUBSTITUTED CYCLOHEXANOLS AUSPEX PHARMACEUTICALS, INC. (US) 2009-01-29 US claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007135574-A1 USE OF PARASYMPATHOLYTIC SUBSTANCES TO ENHANCE AND ACCELERATE STEM CELL DIFFERENTIATION, RELATED METHOD AND COMPOSITIONS UNIVERSITA' DEGLI STUDI DI TORINO (IT) 2007-11-29 WO claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
EP-1273301-B1 Pharmaceutical preparations based on active ingredients susceptible to illicit administration ALTERGON SA (CH) 2006-09-06 EP claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10689370-B2 Cyclopropane carboxamide modulators of cystic fibrosis transmembrane conductance regulator CFTR, CLCN2, TMEM120A CYP2D6 4330/4885CYP3A4 4062/4885CYP1A2 4452/4885
US-20090028873-A1 SUBSTITUTED CYCLOHEXANOLS OPRM1, OPRD1, OPRK1 CYP2D6 57/4885CYP3A4 162/4885CYP1A2 35/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.