SCHEMBL24914458

SCHEMBL24914458

CC(C)(C)OC(=O)N1CCc2c(c(=O)[nH]c3ccccc23)C1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MTHFD2 P13995 1/20 0.60
TRPV1 Q8NER1 6/20 0.53
FAAH O00519 3/20 0.51
LMNA P02545 1/20 0.50
MAPT P10636 1/20 0.50
BAZ2B Q9UIF8 1/20 0.50
F12 P00748 3/20 0.48
MAPK1 P28482 1/20 0.46
ADRA2A P08913 1/20 0.45
ADRA1A P35348 1/20 0.45
GPX4 P36969 1/20 0.45
DDB1 Q16531 1/20 0.44
CRBN Q96SW2 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
PARP1 P09874 1/20 0.44
TNKS2 Q9H2K2 1/20 0.44
PARP2 Q9UGN5 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2241936 0.86 MAPT (0.69) TRPV1FAAHLMNAMAPTBAZ2B
SCHEMBL350201 0.86 TRPV1 (0.69) TRPV1FAAHLMNAMAPTBAZ2B
SCHEMBL29357331 0.86 MAPT (0.69) TRPV1FAAHLMNAMAPTBAZ2B
SCHEMBL32660187 0.84 ESR2 (0.46) MTHFD2BAZ2BF12PARP1TNKS2
SCHEMBL31164770 0.84 ESR2 (0.46) MTHFD2BAZ2BF12PARP1TNKS2
SCHEMBL24914461 0.84 ADORA1 (0.43) MTHFD2TRPV1MAPTF12MAPK1
Acetic Acid SCHEMBL8718251 0.83 TRPV1 (0.68) TRPV1FAAHLMNAMAPTBAZ2B
Acetic Acid SCHEMBL8714196 0.83 MAPT (0.68) TRPV1FAAHLMNAMAPTBAZ2B
SCHEMBL24914511 0.83 MTHFD2 (0.41) MTHFD2TRPV1MAPTF12MAPK1
SCHEMBL24914388 0.82 DDB1 (0.52) MTHFD2MAPTF12MAPK1DDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023284807-A1 COMPOUND CONTAINING TETRAHYDRONAPHTHYRIDONE OR TETRAHYDROPYRIDOPYRIMIDINONE SKELETON, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL USE THEREOF 中国药科大学 2023-01-19 WO disclosed