SCHEMBL24914388

SCHEMBL24914388

CC(C)(C)OC(=O)N1CCc2c(c(=O)[nH]c3ncccc23)C1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.52
CRBN Q96SW2 1/20 0.52
DTYMK P23919 1/20 0.45
KIT P10721 2/20 0.44
PARP1 P09874 1/20 0.43
TNKS2 Q9H2K2 1/20 0.43
PARP2 Q9UGN5 1/20 0.43
POLB P06746 1/20 0.43
MAPT P10636 2/20 0.43
MAPK1 P28482 1/20 0.42
C5AR1 P21730 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
GRM5 P41594 1/20 0.41
F12 P00748 3/20 0.41
MTHFD2 P13995 1/20 0.41
MKNK1 Q9BUB5 2/20 0.41
CCNK O75909 1/20 0.41
CDK12 Q9NYV4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL46600 0.87 DDB1 (0.49) DDB1CRBNDTYMKKITPARP1
SCHEMBL30339672 0.84 KIT (0.48) DDB1CRBNDTYMKKITPOLB
SCHEMBL24101723 0.84 KIT (0.48) DDB1CRBNDTYMKKITPOLB
SCHEMBL31119374 0.83 MTHFD2 (0.49) PARP1MTHFD2
SCHEMBL24914501 0.83 KIT (0.42) DDB1CRBNKITPARP1TNKS2
SCHEMBL24914458 0.82 MTHFD2 (0.60) DDB1CRBNPARP1TNKS2PARP2
SCHEMBL2485934 0.81 MKNK1 (0.46) DDB1CRBNPARP1TNKS2PARP2
SCHEMBL2484902 0.79 MKNK1 (0.46) DDB1CRBNPARP1TNKS2PARP2
SCHEMBL23580395 0.78 ESR2 (0.42) DDB1CRBNPARP1TNKS2PARP2
SCHEMBL24914504 0.77 MKNK1 (0.42) DDB1CRBNPARP1TNKS2PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260022123-A1 Methods of Making Modified BTK Inhibitors PRINCIPIA BIOPHARMA INC. (US) 2026-01-22 US disclosed
WO-2025217420-A1 PYRIDINONE COMPOUNDS, METHODS AND USES THEREOF ZENO MANAGEMENT, INC. (US) 2025-10-16 WO disclosed
CN-115677719-B Aryl heterocyclic compound and preparation method and application thereof 复旦大学 2025-03-07 CN disclosed
CN-119343340-A Methods of preparing modified BTK inhibitors 普林斯匹亚生物制药公司 2025-01-21 CN disclosed
US-20240327408-A1 COMPOUNDS CONTAINING TETRAHYDRONAPHTHYRIDINONE OR TETRAHYDROPYRIDOPYRIMIDINONE SKELETON, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USE THEREOF CHINA PHARMACEUTICAL UNIVERSITY (CN) 2024-10-03 US disclosed
WO-2024088109-A1 ARYL HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF 复旦大学 2024-05-02 WO disclosed
CN-115960074-A Fluorine-containing ferroelectric liquid crystal molecules containing heteroatom hexatomic alicyclic ring and synthesis method thereof 华南理工大学 2023-04-14 CN disclosed
WO-2023284807-A1 COMPOUND CONTAINING TETRAHYDRONAPHTHYRIDONE OR TETRAHYDROPYRIDOPYRIMIDINONE SKELETON, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL USE THEREOF 中国药科大学 2023-01-19 WO disclosed
WO-2023284807-A1 COMPOUND CONTAINING TETRAHYDRONAPHTHYRIDONE OR TETRAHYDROPYRIDOPYRIMIDINONE SKELETON, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL USE THEREOF 中国药科大学 2023-01-19 WO disclosed
CN-115611896-A Compound containing tetralone or tetrahydropyridopyrimidone skeleton and preparation method and pharmaceutical application thereof 中国药科大学 2023-01-17 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260022123-A1 Methods of Making Modified BTK Inhibitors BTK, TEC, SYK DDB1 2030/4885CRBN 1630/4885DTYMK 400/4885
US-20240327408-A1 COMPOUNDS CONTAINING TETRAHYDRONAPHTHYRIDINONE OR TETRAHYDROPYRIDOPYRIMIDINONE SKELETON, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USE THEREOF PRCP, TMPRSS15, WEE1 DDB1 3529/4885CRBN 1365/4885DTYMK 2632/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.