SCHEMBL24914501

SCHEMBL24914501

CC(C)(C)OC(=O)N1CCc2c(c(=O)[nH]c3ncncc23)C1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KIT P10721 2/20 0.42
F12 P00748 3/20 0.41
MKNK1 Q9BUB5 2/20 0.41
ADORA1 P30542 1/20 0.40
MAPT P10636 3/20 0.40
DDB1 Q16531 2/20 0.40
CRBN Q96SW2 2/20 0.40
NR1H2 P55055 1/20 0.40
PARP1 P09874 1/20 0.39
TNKS2 Q9H2K2 1/20 0.39
PARP2 Q9UGN5 1/20 0.39
ESR2 Q92731 1/20 0.38
C5AR1 P21730 1/20 0.38
SPR P35270 1/20 0.38
KDM4E B2RXH2 1/20 0.38
SCN9A Q15858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24914388 0.83 DDB1 (0.52) KITF12MKNK1MAPTDDB1
SCHEMBL23580395 0.78 ESR2 (0.42) F12MKNK1ADORA1DDB1CRBN
SCHEMBL24914504 0.77 MKNK1 (0.42) MKNK1ADORA1MAPTDDB1CRBN
SCHEMBL24914458 0.76 MTHFD2 (0.60) F12MAPTDDB1CRBNPARP1
SCHEMBL24914461 0.76 ADORA1 (0.43) F12ADORA1MAPTDDB1CRBN
SCHEMBL2485934 0.75 MKNK1 (0.46) MKNK1MAPTDDB1CRBNNR1H2
SCHEMBL24914511 0.75 MTHFD2 (0.41) F12ADORA1MAPTDDB1CRBN
SCHEMBL24914515 0.74 NR1H2 (0.44) F12MKNK1ADORA1MAPTDDB1
SCHEMBL30879376 0.74 MKNK1 (0.55) MKNK1ADORA1MAPTKDM4E
SCHEMBL23580642 0.74 ESR2 (0.42) F12MKNK1ADORA1DDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023284807-A1 COMPOUND CONTAINING TETRAHYDRONAPHTHYRIDONE OR TETRAHYDROPYRIDOPYRIMIDINONE SKELETON, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL USE THEREOF 中国药科大学 2023-01-19 WO disclosed