SCHEMBL2491468

SCHEMBL2491468

c1ccc2[nH]c([C@@H]3CCC[N]3)nc2c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ABCB11 O95342 1/20 0.43
TP53 P04637 1/20 0.43
PKM P14618 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HTR2B P41595 3/20 0.42
KMT2A Q03164 2/20 0.42
BCHE P06276 2/20 0.41
ACHE P22303 2/20 0.41
MASP2 O00187 1/20 0.41
MEN1 O00255 1/20 0.41
NUDT1 P36639 1/20 0.41
AOC3 Q16853 1/20 0.41
POLB P06746 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5598283 0.95 BCHE (0.43) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL2201109 0.79 KMT2A (0.42) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL2674802 0.76 HTR2B (0.55) NPC1RAB9AKDM4EHTR2BKMT2A
SCHEMBL6756134 0.76 NPC1 (0.59) NPC1RAB9AKDM4EHTR2BKMT2A
SCHEMBL2276872 0.75 ALDH1A1 (0.59) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL3557180 0.75 HTR2B (0.46) NPC1RAB9AKDM4EHTR2BKMT2A
SCHEMBL3124136 0.75 MPO (0.38) NPC1RAB9AALDH1A1KDM4EHSD17B10
SCHEMBL3250003 0.75 MPO (0.38) NPC1RAB9AALDH1A1KDM4EHSD17B10
SCHEMBL6757201 0.75 NPC1 (0.62) NPC1RAB9AKDM4EHTR2BPOLB
SCHEMBL724921 0.75 NPC1 (0.62) NPC1RAB9AKDM4EHTR2BPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379524-A1 SEROTONIN 5-HT2B RECEPTOR INHIBITORS Boehringer Ingelheim International GmbH (DE) 2011-10-26 EP disclosed
WO-2010080357-A1 SEROTONIN 5-HT2B RECEPTOR INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-07-15 WO disclosed