SCHEMBL24920546

SCHEMBL24920546

COCc1ccnc(N2CC(S(C)(=O)=O)C2)n1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.37
NR1H2 P55055 2/20 0.36
GPR119 Q8TDV5 1/20 0.34
CA12 O43570 6/20 0.34
CA1 P00915 6/20 0.34
CA2 P00918 6/20 0.34
CA9 Q16790 6/20 0.34
CTSS P25774 1/20 0.34
HCRTR1 O43613 3/20 0.33
HCRTR2 O43614 3/20 0.33
RXRA P19793 3/20 0.33
GRIN1 Q05586 3/20 0.33
GRIN2B Q13224 3/20 0.33
PTGS2 P35354 1/20 0.33
EGFR P00533 1/20 0.32
NR1H3 Q13133 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24921022 0.82 AOC3 (0.38) AOC3HCRTR1HCRTR2RXRAGRIN1
SCHEMBL24921790 0.81 AOC3 (0.39) AOC3HCRTR1HCRTR2RXRAGRIN1
SCHEMBL24920529 0.80 AOC3 (0.36) AOC3RXRAGRIN1GRIN2BEGFR
SCHEMBL24920547 0.78 AOC3 (0.38) AOC3NR1H2HCRTR1HCRTR2RXRA
SCHEMBL20745925 0.78 AOC3 (0.35) AOC3NR1H2CA12CA1CA2
SCHEMBL24921046 0.77 AOC3 (0.38) AOC3HCRTR1HCRTR2RXRAGRIN1
SCHEMBL24920543 0.77 DYRK1A (0.46) AOC3
SCHEMBL24921023 0.76 AOC3 (0.44) AOC3CA12CA1CA2CA9
SCHEMBL24921040 0.76 AOC3 (0.44) AOC3CA12CA1CA2CA9
SCHEMBL24921025 0.75 RXRA (0.39) AOC3RXRAGRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed