SCHEMBL24920746

SCHEMBL24920746

Cc1ccc(C2(c3ccc(OCc4ccnc(-c5nncs5)n4)cc3)COC2)cc1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.37
RAB9A P51151 5/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
PTGS2 P35354 2/20 0.32
MAPT P10636 1/20 0.32
TSHR P16473 1/20 0.32
HPGD P15428 1/20 0.32
GAA P10253 1/20 0.31
PDE10A Q9Y233 1/20 0.31
F2RL3 Q96RI0 2/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
CASP3 P42574 1/20 0.30
SENP8 Q96LD8 1/20 0.30
SENP7 Q9BQF6 1/20 0.30
SENP6 Q9GZR1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24920863 0.89 NPC1 (0.37) NPC1RAB9ASMN1; SMN2PTGS2MAPT
SCHEMBL24920730 0.83 NPC1 (0.35) NPC1RAB9ASMN1; SMN2MAPTHPGD
SCHEMBL24920743 0.82 NPC1 (0.36) NPC1RAB9ASMN1; SMN2TSHRHPGD
SCHEMBL24920751 0.81 RAB9A (0.47) NPC1RAB9ASMN1; SMN2PTGS2MAPT
SCHEMBL24921649 0.81 NPC1 (0.40) NPC1RAB9ASMN1; SMN2MAPTTSHR
SCHEMBL24920745 0.81 NPC1 (0.35) NPC1RAB9ASMN1; SMN2HPGDGAA
SCHEMBL24920736 0.79 NPC1 (0.34) NPC1RAB9ASMN1; SMN2MAPTTSHR
SCHEMBL24920749 0.79 NPC1 (0.36) NPC1RAB9ASMN1; SMN2MAPTHPGD
SCHEMBL24920723 0.79 NPC1 (0.35) NPC1RAB9ASMN1; SMN2PTGS2MAPT
SCHEMBL24920727 0.78 NPC1 (0.34) NPC1RAB9ASMN1; SMN2MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed