SCHEMBL24920804

SCHEMBL24920804

COc1ncc(F)c(-n2nccn2)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 2/20 0.37
HCRTR2 O43614 1/20 0.34
CYP1A2 P05177 7/20 0.34
TGFBR1 P36897 1/20 0.33
TGFBR2 P37173 1/20 0.33
CYP3A4 P08684 4/20 0.33
MEN1 O00255 2/20 0.33
ALDH1A1 P00352 2/20 0.33
KMT2A Q03164 2/20 0.33
HSD17B10 Q99714 2/20 0.33
GLA P06280 1/20 0.33
HIF1A Q16665 1/20 0.33
TSHR P16473 2/20 0.32
CYP2C19 P33261 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2D6 P10635 1/20 0.32
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
SLC9A1 P19634 2/20 0.32
SLC9A2 Q9UBY0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24920813 0.81 PDK2 (0.37) PDK2CYP1A2CYP3A4MEN1ALDH1A1
SCHEMBL24920808 0.78 ALDH1A1 (0.38) PDK2CYP1A2TGFBR1TGFBR2CYP3A4
SCHEMBL24920900 0.76 PDK2 (0.35) PDK2CYP1A2CYP3A4MEN1ALDH1A1
SCHEMBL21905028 0.71 CYP1A2 (0.37) CYP1A2CYP3A4MEN1ALDH1A1KMT2A
SCHEMBL26258152 0.71 PDK2 (0.39) PDK2HCRTR2CYP1A2CYP3A4MEN1
SCHEMBL24921600 0.70 TAAR1 (0.34) HCRTR2TGFBR2NPC1RAB9AGRIN1
SCHEMBL24920789 0.70 HCRTR2 (0.37) HCRTR2ALDH1A1
SCHEMBL2511301 0.70 QPCT (0.39) CYP1A2CYP3A4MEN1ALDH1A1KMT2A
SCHEMBL14972263 0.70 CYP1A2 (0.45) CYP1A2CYP3A4MEN1ALDH1A1KMT2A
SCHEMBL24921590 0.70 TUBB4A (0.34) CYP1A2ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed