SCHEMBL24920833

SCHEMBL24920833

COc1cnnc(-c2nnc(C)o2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR Q13258 1/20 0.41
NPC1 O15118 5/20 0.37
RAB9A P51151 5/20 0.37
KMT2A Q03164 3/20 0.37
MAPK14 Q16539 2/20 0.34
TLR8 Q9NR97 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
MAPK8 P45983 1/20 0.33
MAPK10 P53779 1/20 0.33
ALDH1A1 P00352 3/20 0.33
MAPT P10636 3/20 0.33
HPGD P15428 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
TP53 P04637 2/20 0.33
MEN1 O00255 1/20 0.33
KDM4E B2RXH2 3/20 0.33
HSD17B10 Q99714 2/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24921172 0.75 CCR1 (0.59) PTGDRNPC1RAB9AKMT2AMAPK14
SCHEMBL24920835 0.75 NOTUM (0.51) KMT2ATLR8ALDH1A1MAPTHPGD
SCHEMBL24920867 0.74 CNR2 (0.37) PTGDRNPC1RAB9AKMT2AMAPT
SCHEMBL12923721 0.73 NPC1 (0.44) PTGDRNPC1RAB9AKMT2AMAPK14
SCHEMBL12923984 0.73 CHRNB2 (0.46) NPC1RAB9AKMT2AMAPK14ALDH1A1
SCHEMBL24920815 0.72 CCR1 (0.34)
SCHEMBL24921142 0.71 GABRG2 (0.44) NPC1RAB9AKMT2AMAPK14TLR8
SCHEMBL24921547 0.71 NPC1 (0.37) PTGDRNPC1RAB9AKMT2AMAPK14
SCHEMBL24920812 0.71 MAPT (0.44) NPC1RAB9AKMT2AALDH1A1MAPT
SCHEMBL24921502 0.70 NPC1 (0.40) PTGDRNPC1RAB9AKMT2AMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed