SCHEMBL24920840

SCHEMBL24920840

COc1cc(-c2nnco2)ncn1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.45
ALDH1A1 P00352 3/20 0.44
HPGD P15428 2/20 0.44
MAPK1 P28482 2/20 0.44
NOTUM Q6P988 10/20 0.43
TSHR P16473 1/20 0.37
CYP2C19 P33261 2/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
HSD17B10 Q99714 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
KMT2A Q03164 1/20 0.35
GAA P10253 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP1A1 P04798 1/20 0.33
CYP1B1 Q16678 1/20 0.33
LMNA P02545 1/20 0.33
NOD2 Q9HC29 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5444260 0.75 RAB9A (0.42) MAPTALDH1A1HPGDNOTUMTSHR
SCHEMBL14031552 0.75 CYP2C19 (0.37) MAPTALDH1A1TSHRCYP2C19NPC1
SCHEMBL24921990 0.75 MAPT (0.42) MAPTALDH1A1HPGDMAPK1NOTUM
SCHEMBL5417649 0.74 NOTUM (0.46) MAPTNOTUMTSHR
SCHEMBL24921991 0.74 ALDH1A1 (0.47) MAPTALDH1A1HPGDMAPK1NOTUM
SCHEMBL24921176 0.73 NOTUM (0.54) MAPTALDH1A1HPGDMAPK1NOTUM
SCHEMBL25693362 0.73 NOTUM (0.44) MAPTALDH1A1HPGDMAPK1NOTUM
SCHEMBL24920826 0.73 CYP2C19 (0.36) ALDH1A1HPGDCYP2C19NPC1RAB9A
SCHEMBL25986790 0.73 TSHR (0.37) MAPTALDH1A1HPGDMAPK1NOTUM
SCHEMBL24920820 0.72 CYP2C19 (0.38) MAPTCYP2C19NPC1RAB9ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed