SCHEMBL24921997

SCHEMBL24921997

COc1cnc(-n2ncc(C)n2)cn1

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 1/20 0.35
PDE10A Q9Y233 1/20 0.33
FGFR1 P11362 1/20 0.31
FGFR4 P22455 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24921539 0.78 SIRT6 (0.39) SIRT6
SCHEMBL24921589 0.78 MEN1 (0.44)
SCHEMBL24920819 0.77 CYP2C19 (0.45) PDE10A
SCHEMBL24921560 0.76 EGLN1 (0.37) PDE10A
SCHEMBL24921989 0.76 KDM4E (0.37) PDE10A
SCHEMBL24920811 0.75 PIK3CG (0.34) PDE10A
SCHEMBL24921968 0.75 PDE10A (0.37) PDE10A
SCHEMBL24922002 0.75 MEN1 (0.30)
SCHEMBL24921165 0.73 ALOX5 (0.40) PDE10A
SCHEMBL24921999 0.71 OGA (0.33) PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed