SCHEMBL24933354

SCHEMBL24933354

CC(C)(C)OC(=O)N[C@H]1C[C@H](COc2ccc(-c3cc(C(N)=O)c(=O)[nH]c3C(F)(F)F)cc2)C1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 2/20 0.36
HSD17B1 P14061 5/20 0.36
HSD17B2 P37059 5/20 0.36
PARP1 P09874 4/20 0.36
SCN9A Q15858 1/20 0.35
KAT8 Q9H7Z6 1/20 0.34
PARP2 Q9UGN5 1/20 0.34
ACACB O00763 1/20 0.34
PARP15 Q460N3 1/20 0.33
PARP10 Q53GL7 1/20 0.33
BTK Q06187 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24933255 0.83 CHEK2 (0.47) CHEK2
SCHEMBL24933356 0.81 PARP10 (0.52) CHEK2PARP2PARP15PARP10FFAR4
SCHEMBL24933017 0.81 PRKAB2 (0.42) CHEK2HSD17B1HSD17B2PARP2PARP15
SCHEMBL24933399 0.80 CHEK2 (0.52) CHEK2SCN9A
SCHEMBL24933633 0.80 PARP10 (0.53) CHEK2PARP2PARP15PARP10FFAR4
SCHEMBL24933494 0.80 IRAK4 (0.41) CHEK2HSD17B1HSD17B2PARP2PARP15
SCHEMBL24933789 0.79 CHEK2 (0.42) CHEK2PARP2PARP15PARP10
SCHEMBL24933589 0.79 XDH (0.49) CHEK2HSD17B1HSD17B2PARP1PARP2
SCHEMBL24932946 0.79 XDH (0.42) CHEK2HSD17B1HSD17B2PARP2PARP15
SCHEMBL24932956 0.77 FYN (0.45) CHEK2HSD17B1HSD17B2PARP1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed