SCHEMBL24933588

SCHEMBL24933588

CS(=O)(=O)Nc1ccc(-c2cc(C(N)=O)c(=O)[nH]c2C(F)(F)F)cc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHUK O15111 6/20 0.49
IKBKB O14920 5/20 0.49
KIF11 P52732 4/20 0.45
INSR P06213 1/20 0.44
MAPK8 P45983 1/20 0.44
CAMKK2 Q96RR4 1/20 0.44
HSD17B1 P14061 4/20 0.41
HSD17B2 P37059 4/20 0.41
PTGS2 P35354 1/20 0.40
BRD4 O60885 2/20 0.40
CSF1R P07333 1/20 0.39
CHEK2 O96017 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24933208 0.84 KMT2A (0.40) KIF11HSD17B1HSD17B2BRD4
SCHEMBL30240693 0.82 MAOB (0.41) CHUKIKBKBKIF11INSRMAPK8
SCHEMBL24933359 0.82 HSD17B2 (0.50) HSD17B1HSD17B2
SCHEMBL24933312 0.80 BTK (0.42) CHUKIKBKBMAPK8HSD17B1HSD17B2
SCHEMBL24933605 0.80 HSD17B2 (0.41) KIF11HSD17B1HSD17B2
SCHEMBL24933339 0.79 HSD17B1 (0.41) HSD17B1HSD17B2CHEK2
SCHEMBL24933182 0.79 HSD17B1 (0.44) HSD17B1HSD17B2CHEK2
SCHEMBL24932950 0.79 HSD17B2 (0.52) CHUKIKBKBHSD17B1HSD17B2BRD4
SCHEMBL24933053 0.79 KDM4E (0.44) HSD17B1HSD17B2PTGS2
SCHEMBL24933771 0.78 IKBKB (0.42) CHUKIKBKBKIF11HSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4373809-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2024-05-29 EP claimed
CN-117980292-A Substituted pyridone compounds for the treatment of orthomyxoviral infections 诺华股份有限公司 2024-05-03 CN claimed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO claimed
EP-4373809-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2024-05-29 EP disclosed
CN-117980292-A Substituted pyridone compounds for the treatment of orthomyxoviral infections 诺华股份有限公司 2024-05-03 CN disclosed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed