SCHEMBL24933339

SCHEMBL24933339

NC(=O)c1cc(-c2ccc(I)cc2)c(C(F)(F)F)[nH]c1=O

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 11/20 0.41
HSD17B2 P37059 11/20 0.41
PARP1 P09874 3/20 0.33
MAP2K2 P36507 1/20 0.33
MAP2K1 Q02750 1/20 0.33
CASP1 P29466 1/20 0.33
CDC7 O00311 1/20 0.33
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
BTK Q06187 1/20 0.32
CHEK2 O96017 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24933605 0.88 HSD17B2 (0.41) HSD17B1HSD17B2PARP1CASP1
SCHEMBL24933312 0.88 BTK (0.42) HSD17B1HSD17B2CDC7CDK5BTK
SCHEMBL24933359 0.86 HSD17B2 (0.50) HSD17B1HSD17B2CDC7BTK
SCHEMBL24932950 0.86 HSD17B2 (0.52) HSD17B1HSD17B2PARP1CDC7
SCHEMBL24933771 0.85 IKBKB (0.42) HSD17B1HSD17B2PARP1CDK5CDK5R1
SCHEMBL24933343 0.84 HSD17B1 (0.39) HSD17B1HSD17B2PARP1CASP1CDK5
SCHEMBL24933053 0.83 KDM4E (0.44) HSD17B1HSD17B2PARP1CASP1CDC7
SCHEMBL24933181 0.82 HSD17B2 (0.41) HSD17B1HSD17B2PARP1CDK5CDK5R1
SCHEMBL24933333 0.81 GSTP1 (0.44) HSD17B1HSD17B2BTKCHEK2
SCHEMBL24933182 0.81 HSD17B1 (0.44) HSD17B1HSD17B2BTKCHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed