SCHEMBL24933693

SCHEMBL24933693

Cc1nc(C)c(COc2ccc(-c3cc(C(N)=O)c(=O)[nH]c3C(F)(F)F)cc2)s1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 15/20 0.44
PPARA Q07869 9/20 0.44
PPARG P37231 6/20 0.44
FFAR1 O14842 9/20 0.41
HSD17B1 P14061 1/20 0.38
HSD17B2 P37059 1/20 0.38
CHRM5 P08912 1/20 0.37
SLC6A3 Q01959 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24933849 0.87 HSD17B1 (0.39) PPARDPPARAPPARGFFAR1HSD17B1
SCHEMBL24933254 0.85 HSD17B1 (0.38) PPARDPPARAPPARGFFAR1HSD17B1
SCHEMBL24933002 0.84 HSD17B1 (0.38) HSD17B1HSD17B2
SCHEMBL24933706 0.83 PARP10 (0.39) PPARDPPARAPPARGHSD17B1HSD17B2
SCHEMBL24933809 0.83 HSD17B1 (0.38) PPARDHSD17B1HSD17B2
SCHEMBL24933881 0.81 HSD17B1 (0.38) PPARDHSD17B1HSD17B2
SCHEMBL24933639 0.81 NMT1 (0.40) FFAR1HSD17B1HSD17B2
SCHEMBL30240787 0.81 HSD17B1 (0.38) PPARDHSD17B1HSD17B2
SCHEMBL24933369 0.81 HSD17B1 (0.38) PPARDHSD17B1HSD17B2
SCHEMBL30240751 0.80 HSD17B1 (0.41) HSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4373809-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2024-05-29 EP claimed
CN-117980292-A Substituted pyridone compounds for the treatment of orthomyxoviral infections 诺华股份有限公司 2024-05-03 CN claimed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO claimed
EP-4373809-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2024-05-29 EP disclosed
CN-117980292-A Substituted pyridone compounds for the treatment of orthomyxoviral infections 诺华股份有限公司 2024-05-03 CN disclosed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed