SCHEMBL24933729

SCHEMBL24933729

NC(=O)c1cc(-c2ccc(OCc3cnc(NC4CCOC4)nc3)cc2)c(C(F)(F)F)[nH]c1=O

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.36
RAB9A P51151 1/20 0.35
MAPK8 P45983 1/20 0.35
MAPK9 P45984 1/20 0.35
SYK P43405 4/20 0.35
MAPK1 P28482 3/20 0.35
MAPK3 P27361 1/20 0.35
PDPK1 O15530 1/20 0.34
XDH P47989 1/20 0.34
HSD17B1 P14061 3/20 0.33
HSD17B2 P37059 3/20 0.33
EGLN1 Q9GZT9 3/20 0.33
JAK2 O60674 1/20 0.33
CHEK1 O14757 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24933234 0.94 HSD17B1 (0.35) SYKPDPK1HSD17B1HSD17B2CHEK1
SCHEMBL24932987 0.91 SYK (0.40) MAPK8SYKPDPK1HSD17B1HSD17B2
SCHEMBL24933812 0.90 SYK (0.39) MAPK8SYKPDPK1JAK2CHEK1
SCHEMBL24933228 0.85 CYP11B1 (0.37) ACACBSYKXDHHSD17B1HSD17B2
SCHEMBL24933678 0.85 XDH (0.44) XDH
SCHEMBL24932967 0.83 FFAR1 (0.36) SYKHSD17B1HSD17B2JAK2
SCHEMBL24933810 0.83 FFAR4 (0.40) HSD17B1HSD17B2
SCHEMBL24933216 0.83 HSD17B1 (0.36) MAPK8HSD17B1HSD17B2
SCHEMBL30240717 0.81 CYP11B2 (0.38) MAPK1XDHHSD17B1HSD17B2
SCHEMBL24932983 0.81 SCN9A (0.39) SYKHSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4373809-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2024-05-29 EP claimed
CN-117980292-A Substituted pyridone compounds for the treatment of orthomyxoviral infections 诺华股份有限公司 2024-05-03 CN claimed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO claimed
EP-4373809-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2024-05-29 EP disclosed
CN-117980292-A Substituted pyridone compounds for the treatment of orthomyxoviral infections 诺华股份有限公司 2024-05-03 CN disclosed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed