Metaterol

Metaterol

SCHEMBL249460

CC(C)NCC(O)c1cccc(O)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 6/20 0.70
ADRB2 P07550 5/20 0.70
TSHR P16473 5/20 0.70
ADRB1 P08588 4/20 0.70
ADRA1A P35348 3/20 0.70
ADRB3 P13945 3/20 0.70
NFKB1 P19838 2/20 0.70
ADRA1B P35368 2/20 0.70
DRD3 P35462 2/20 0.70
HTR1A P08908 1/20 0.70
ADRA2A P08913 1/20 0.70
ADRA2B P18089 1/20 0.70
ADRA2C P18825 1/20 0.70
DRD1 P21728 1/20 0.70
HTR7 P34969 1/20 0.70
RAB9A P51151 1/20 0.70
SLC6A3 Q01959 1/20 0.70
LMNA P02545 4/20 0.68
KDM4E B2RXH2 3/20 0.68
BLM P54132 3/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Metaterol SCHEMBL10614404 0.98 HIF1A (0.71) HIF1AADRB2TSHRADRB1ADRA1A
Metaproterenol SCHEMBL1679992 0.90 ADRB2 (0.75) HIF1AADRB2TSHRADRB1ADRA1A
SCHEMBL4625692 0.85 ADRB2 (0.64) HIF1AADRB2TSHRADRB1ADRA1A
Metaproterenol SCHEMBL15163491 0.83 ADRB2 (0.67) HIF1AADRB2TSHRADRB1ADRA1A
SCHEMBL31676604 0.83 HIF1A (0.61) HIF1AADRB2TSHRADRB1ADRA1A
SCHEMBL22362712 0.83 HIF1A (0.61) HIF1AADRB2TSHRADRB1ADRA1A
SCHEMBL20819520 0.83 HIF1A (0.61) HIF1AADRB2TSHRADRB1ADRA1A
SCHEMBL20819521 0.83 HIF1A (0.61) HIF1AADRB2TSHRADRB1ADRA1A
SCHEMBL31676571 0.83 HIF1A (0.61) HIF1AADRB2TSHRADRB1ADRA1A
SCHEMBL19329958 0.83 HIF1A (0.61) HIF1AADRB2TSHRADRB1ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
US-4407819-A ANIMAL GROWTH REGULATORS AMERICAN CYANAMID COMPANY (US) 1983-10-04 US claimed
CN-114057590-A Synthetic method of key intermediate of odaterol 安徽有吉医药科技有限公司 2022-02-18 CN disclosed
US-20220031719-A1 ANTIVIRAL THERAPEUTIC DRUG COMBINATIONS THE UNIVERSITY OF TULSA (US) 2022-02-03 US disclosed
CN-111574529-A Muscarinic receptor M3 antagonists and β 2-adrenergic receptor agonist bridged ring derivatives 四川海思科制药有限公司 2020-08-25 CN disclosed
EP-2401275-B1 NAPHTHYRIDINE DERIVATIVES HAVING BRONCHODILATING ACTIVITY RESPIRATORIUS AB (SE) 2013-07-24 EP disclosed
US-8454582-B2 Methods and devices for the treatment of ocular conditions SURMODICS, INC. (US) 2013-06-04 US disclosed
US-8415333-B2 Bronchodilating diazaheteroaryls RESPIRATORIOUS AB (SE) 2013-04-09 US disclosed
US-20120040942-A1 NOVEL BRONCHODILATING DIAZAHETEROARYLS RESPIRATORIUS AB (SE) 2012-02-16 US disclosed
EP-2401275-A1 NOVEL BRONCHODILATING DIAZAHETEROARYLS Respiratorius AB (SE) 2012-01-04 EP disclosed
US-20110159073-A1 METHODS AND DEVICES FOR THE TREATMENT OF OCULAR CONDITIONS DEJUAN EUGENE 2011-06-30 US disclosed
US-6261537-B1 TARGETS AND ULTRASOUND DIAGNOSIS OF ACTIVE MATERIALS, AQUEOUS CARRIER LIQUIDS, CARRIERS AND FILM FORMING SURFACTANT PHOSPHATIDES NYCOMED IMAGING AS (NO) 2001-07-17 US disclosed
EP-1086947-A1 Somatostatin antagonists and agonists that act at the SST subtype 2 receptor Pfizer Products Inc. (US) 2001-03-28 EP disclosed
US-4754047-A ANIMAL GROWTH REGULATORS AMERICAN CYANAMID COMPANY (US) 1988-06-28 US disclosed
US-4522822-A Phenylethane derivatives and acid addition salts thereof for increasing lean meat deposition and/or improving lean meat to fat ratio in warm blooded animals AMERICAN CYANAMID COMPANY (US) 1985-06-11 US disclosed
US-4501751-A Phenylethanolamine derivatives and acid addition salts thereof for enhancing the growth rate of meat-producing animals and improving the efficiency of feed utilization thereby AMERICAN CYANAMID COMPANY (US) 1985-02-26 US disclosed
EP-0026298-B1 METHOD FOR PROMOTING GROWTH AND REDUCING FAT IN ANIMALS USING PHENYLETHANOLAMINE DERIVATIVES AMERICAN CYANAMID COMPANY (US) 1984-04-18 EP disclosed
US-4407819-A ANIMAL GROWTH REGULATORS AMERICAN CYANAMID COMPANY (US) 1983-10-04 US disclosed
US-4404222-A Phenylethanolamine derivatives and acid addition salts thereof for enhancing the growth rate of meat-producing animals and improving the efficiency of feed utilization thereby AMERICAN CYANAMID COMPANY (US) 1983-09-13 US disclosed
EP-0026298-A1 Method for promoting growth and reducing fat in animals using phenylethanolamine derivatives AMERICAN CYANAMID COMPANY (US) 1981-04-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220031719-A1 ANTIVIRAL THERAPEUTIC DRUG COMBINATIONS HK2, G6PD, GCK HIF1A 136/4885ADRB2 2308/4885TSHR 4647/4885
US-20120040942-A1 NOVEL BRONCHODILATING DIAZAHETEROARYLS CHRM3, ADRB1, ADRB3 HIF1A 907/4885ADRB2 5/4885TSHR 1779/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.